SCHEMBL1701229

SCHEMBL1701229

Cc1c(-c2ccco2)n[nH]c1-c1ccc(N)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.40
ADORA2A P29274 5/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2B P29275 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
PDE10A Q9Y233 1/20 0.38
TAAR1 Q96RJ0 1/20 0.36
PDGFRB P09619 1/20 0.36
KIT P10721 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
KDM4E B2RXH2 4/20 0.36
HSD17B10 Q99714 3/20 0.36
USP2 O75604 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592508 0.84 TAAR1 (0.51) PDPK1ADORA2AADORA1ADORA2BHSP90AA1
SCHEMBL1701865 0.76 FYN (0.43) PDGFRBKITCDK5CDK5R1KDM4E
SCHEMBL3059958 0.75 TAAR1 (0.57) PDPK1ADORA2ATAAR1KDM4EHSD17B10
SCHEMBL10305768 0.74 ADORA2A (0.49) PDPK1ADORA2AADORA1ADORA2BHSP90AA1
SCHEMBL27651185 0.66 KDM4E (0.47) ADORA2AADORA1ADORA2BHSP90AA1HSP90AB1
SCHEMBL27671102 0.66 MAPT (0.43) PDPK1ADORA2AADORA1ADORA2BTAAR1
SCHEMBL1701209 0.65 HSP90AA1 (0.48) PDPK1ADORA2AADORA1ADORA2BHSP90AA1
SCHEMBL27203335 0.65 MAPT (0.43) ADORA2AADORA1HSP90AA1HSP90AB1PDE10A
SCHEMBL27512201 0.65 KDM4E (0.50) PDPK1ADORA2AADORA1ADORA2BHSP90AA1
SCHEMBL1701227 0.64 PTGS1 (0.42) ADORA2AADORA1ADORA2BTAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563776-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2011139489-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-11-10 WO disclosed