SCHEMBL2593510

SCHEMBL2593510

C[C@H]1CCC[N+]1(c1ccc2c(c1)CCN(C1CCOCC1)C2=O)[C@H]1CCNC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.42
HRH3 Q9Y5N1 4/20 0.39
HTR2C P28335 12/20 0.37
HTR2B P41595 12/20 0.37
HTR2A P28223 11/20 0.37
MAOA P21397 2/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2595539 0.81 HRH3 (0.37) HRH3
Hydrochloric Acid SCHEMBL2593507 0.80 HRH3 (0.37) HRH3
SCHEMBL2595527 0.76 KEAP1 (0.38)
SCHEMBL2596377 0.72 HRH3 (0.36) HRH3HTR2CHTR2BHTR2A
SCHEMBL14776067 0.72 F10 (0.36)
SCHEMBL2593506 0.71 HRH3 (0.38) HRH3
SCHEMBL2596374 0.71 MCHR1 (0.35) HRH3HTR2CHTR2B
SCHEMBL2595666 0.71 ASIC3 (0.37) HRH3HTR2CHTR2BHTR2AMAOB
SCHEMBL2475614 0.69 HRH3 (0.42) HRH3
SCHEMBL2590061 0.69 HRH3 (0.43) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569303-A1 SUBSTITUTED N-ALKYL AND N-ACYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI (FR) 2013-03-20 EP claimed
WO-2011143145-A1 SUBSTITUTED N-ALKYL AND N-ACYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI (FR) 2011-11-17 WO claimed
EP-2569303-A1 SUBSTITUTED N-ALKYL AND N-ACYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI (FR) 2013-03-20 EP disclosed
WO-2011143145-A1 SUBSTITUTED N-ALKYL AND N-ACYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI (FR) 2011-11-17 WO disclosed