SCHEMBL25947747

SCHEMBL25947747

CNc1cccn(Cc2nc3cccc(COc4ccc(F)cc4F)c3s2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.43
DCPS Q96C86 1/20 0.43
MAP4K1 Q92918 8/20 0.40
MAPK14 Q16539 4/20 0.38
PTGER3 P43115 4/20 0.38
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31304006 0.88 DHFR (0.50) DHFRDCPSMAP4K1MAPK14KDM4E
SCHEMBL21684178 0.88 DHFR (0.50) DHFRDCPSMAP4K1MAPK14KDM4E
SCHEMBL21684767 0.84 ALDH1A1 (0.47) DHFRDCPSMAP4K1MAPK14MEN1
SCHEMBL21702983 0.83 MAPK14 (0.44) MAP4K1MAPK14PSEN1PSEN2APH1B
SCHEMBL25947417 0.81 MAPK14 (0.43) MAP4K1MAPK14PSEN1PSEN2APH1B
SCHEMBL21684882 0.78 MAPK14 (0.47) DHFRDCPSMAP4K1MAPK14
SCHEMBL21683581 0.78 MAP4K1 (0.66) MAP4K1
SCHEMBL21683584 0.78 MAP4K1 (0.66) MAP4K1
SCHEMBL28581797 0.77 MAP4K1 (0.59) MAP4K1
SCHEMBL31450621 0.77 MAP4K1 (0.59) MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4219460-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS Sitari Pharma, Inc. (US) 2023-08-02 EP disclosed