SCHEMBL25948366

SCHEMBL25948366

COC(=O)c1cc2cc(Oc3ccc(N)cc3)c(Br)cc2s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN2 P17706 2/20 0.46
CCNC P24863 1/20 0.45
CDK8 P49336 1/20 0.45
STING1 Q86WV6 6/20 0.43
ICAM1 P05362 3/20 0.42
SELE P16581 3/20 0.42
VCAM1 P19320 2/20 0.42
HDAC1 Q13547 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
CLK1 P49759 3/20 0.38
DYRK1A Q13627 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25948367 0.88 CCNC (0.58) PTPN2CCNCCDK8STING1ICAM1
SCHEMBL29636388 0.81 STING1 (0.61) PTPN2STING1HDAC1HDAC3HDAC4
SCHEMBL20022239 0.81 STING1 (0.61) PTPN2STING1HDAC1HDAC3HDAC4
SCHEMBL16396262 0.78 PTPN2 (0.55) PTPN2STING1HDAC1HDAC3HDAC4
SCHEMBL25948368 0.77 CCNC (0.56) PTPN2CCNCCDK8STING1ICAM1
SCHEMBL20563177 0.75 STING1 (0.61) PTPN2STING1HDAC1HDAC3HDAC4
SCHEMBL20338887 0.75 PTPN2 (0.53) PTPN2STING1HDAC1HDAC3HDAC4
SCHEMBL100069 0.75 MAPT (0.52) PTPN2HDAC1CLK1DYRK1ADYRK1B
SCHEMBL999671 0.75 HDAC1 (0.56) PTPN2HDAC1HDAC3HDAC4HDAC7
SCHEMBL13735896 0.72 PTPN2 (0.59) PTPN2STING1HDAC1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed