SCHEMBL25948854

SCHEMBL25948854

Cc1cc(C)c2ccc(C)n2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
RAPGEF4 Q8WZA2 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
KMT2A Q03164 1/20 0.34
AGER Q15109 1/20 0.34
ESR2 Q92731 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TNKS O95271 4/20 0.32
PARP1 P09874 4/20 0.32
TNKS2 Q9H2K2 4/20 0.32
ADORA3 P0DMS8 1/20 0.32
SLC6A3 Q01959 1/20 0.32
PARP6 Q2NL67 1/20 0.32
PARP10 Q53GL7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24103207 0.71 KDM4E (0.31) FNTAFNTBKDM4EMAPT
SCHEMBL8404416 0.67 SSTR4 (0.38) KDM4EMAPTHSD17B10NPSR1
SCHEMBL7169099 0.65 CHRNA7 (0.38) KDM4EMEN1MAPTALOX15CASP1
SCHEMBL8404413 0.65 KDM4E (0.39) KDM4EMEN1MAPTALOX15CASP1
SCHEMBL25948851 0.64 PTPN1 (0.37) KDM4EMAPTTNKSPARP1TNKS2
SCHEMBL25948856 0.62 NOS3 (0.34) RAPGEF4
SCHEMBL23589214 0.62 EGFR (0.37) RAPGEF4MEN1KMT2AHSD17B10
SCHEMBL8404406 0.62 PTPN1 (0.39) KDM4EMAPTHSD17B10PARP1
SCHEMBL8404415 0.60 KDM4E (0.43) KDM4EMAPTNPSR1
SCHEMBL10889966 0.60 MYC (0.44) RAPGEF4KDM4EMEN1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242533-A9 SUBSTITUTED FUSED HETEROAROMATIC BICYCLIC COMPOUNDS AS KINASE INHIBITORS AND THE USE THEREOF Impact Therapeutics (Shanghai), Inc (CN) 2023-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242533-A9 SUBSTITUTED FUSED HETEROAROMATIC BICYCLIC COMPOUNDS AS KINASE INHIBITORS AND THE USE THEREOF ATR, CHEK1, CHEK2 FNTA 2938/4885FNTB 2490/4885RAPGEF4 1329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.