SCHEMBL2595294

SCHEMBL2595294

NNC(=O)C1CCCCC1c1noc(CO)c1CO

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.31
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2579822 0.76 SMYD3 (0.32)
SCHEMBL2595492 0.75 SMN1; SMN2 (0.36) KCNQ3KCNQ2
SCHEMBL2596228 0.73 SMN1; SMN2 (0.35)
SCHEMBL2593232 0.73 SMN1; SMN2 (0.41)
SCHEMBL2596210 0.73 SMN1; SMN2 (0.35)
SCHEMBL2595298 0.67 SMN1; SMN2 (0.36) KCNQ3KCNQ2
SCHEMBL2596227 0.65 SMN1; SMN2 (0.35)
SCHEMBL29250547 0.64 ALDH1A1 (0.45)
SCHEMBL3623530 0.64 ALDH1A1 (0.45)
SCHEMBL2580221 0.63 TP53 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-20 EP disclosed
WO-2011141396-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-17 WO disclosed