SCHEMBL25958488

SCHEMBL25958488

N=Cc1cnc(C(=O)N2CC3CCC(C3)C2)cc1N

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 7/20 0.37
DPP4 P27487 1/20 0.34
HPGD P15428 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GRM1 Q13255 1/20 0.32
TRPC6 Q9Y210 2/20 0.32
CHRNA7 P36544 2/20 0.32
VNN1 O95497 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25958496 0.81 TRPC6 (0.39) TRPC6
SCHEMBL25958444 0.79 CNR1 (0.43) DPP4HPGDALDH1A1TRPC6
SCHEMBL25958594 0.77 SCN9A (0.40) TRPC6
SCHEMBL25958476 0.75 DPP4 (0.32) DPP4TRPC6
SCHEMBL25958553 0.75 VNN1 (0.43) DPP4HPGDALDH1A1VNN1
SCHEMBL25958544 0.74 VNN1 (0.39) TRPC6VNN1
SCHEMBL25958460 0.73 SMN1; SMN2 (0.46) HPGDALDH1A1VNN1
SCHEMBL25958568 0.69 SMN1; SMN2 (0.37) HPGDVNN1
SCHEMBL24086956 0.68 CHRNA4 (0.40) CHRNA4DPP4CHRNB2CHRNB4CHRNA3
SCHEMBL25958516 0.68 TRPC6 (0.38) ALDH1A1TRPC6VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed