SCHEMBL25969843

SCHEMBL25969843

O=c1c(Cl)c(CO)cnn1Cc1nc(CCc2ccc(C(F)(F)F)cc2)no1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 11/20 0.42
NPBWR1 P48145 1/20 0.39
HTT P42858 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 2/20 0.35
MITF O75030 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NR3C1 P04150 1/20 0.35
FFAR1 O14842 1/20 0.35
PKLR P30613 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25969142 0.89 HTT (0.47) TRPA1HTTRAB9AALDH1A1PKM
SCHEMBL25969149 0.89 TRPA1 (0.52) TRPA1HTTRAB9ANPC1ALDH1A1
SCHEMBL25969147 0.87 ALDH1A1 (0.47) TRPA1NPBWR1HTTRAB9AALDH1A1
SCHEMBL25969061 0.87 TRPA1 (0.44) TRPA1NPBWR1HTTRAB9ANPC1
SCHEMBL25968920 0.80 TRPA1 (0.52) TRPA1
SCHEMBL25969154 0.79 TRPA1 (0.52) TRPA1HTTRAB9ANPC1ALDH1A1
SCHEMBL25970863 0.78 TRPA1 (0.49) TRPA1HTTRAB9ANPC1ALDH1A1
SCHEMBL25970867 0.77 TRPA1 (0.53) TRPA1HTTRAB9ANPC1ALDH1A1
SCHEMBL25969531 0.77 TRPA1 (0.52) TRPA1NPBWR1HTTRAB9ANPC1
SCHEMBL25974095 0.77 TRPA1 (0.55) TRPA1HTTRAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023150591-A2 PYRIDAZINONE COMPOUNDS AS TRPA1 INHIBITORS D.E. SHAW RESEARCH, LLC (US) 2023-08-10 WO disclosed