SCHEMBL25975005

SCHEMBL25975005

CC(C)n1ncc(I)cc1=O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.36
KDM4E B2RXH2 2/20 0.33
TOP2A P11388 1/20 0.31
KMT2A Q03164 1/20 0.31
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30
BPTF Q12830 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20444036 0.78 KMT2A (0.34) HTR3AKDM4ETOP2AKMT2APDE1A
SCHEMBL11287052 0.76 KDM4E (0.33) HTR3AKDM4ETOP2AKMT2APDE1A
SCHEMBL20176157 0.76 KDM4E (0.36) HTR3AKDM4ETOP2AKMT2APDE1A
SCHEMBL12042945 0.65
SCHEMBL19698900 0.65 ADORA2B (0.34) KDM4ETOP2APDE1CBPTF
SCHEMBL1008763 0.65 GCK (0.35) KDM4E
SCHEMBL411297 0.64 ABCB1 (0.41) PDE1APDE1BPDE1C
SCHEMBL6741169 0.64 KMO (0.41) KDM4EPDE1APDE1BPDE1C
SCHEMBL24504750 0.64 DRD4 (0.35)
SCHEMBL16050701 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154282-A1 COMPOUNDS HAVING A T-STRUCTURE FORMED BY AT LEAST FOUR CYCLES FOR USE IN THE TREATMENT OF CANCER AND OTHER INDICATIONS THERAS, INC. (US) 2023-08-17 WO disclosed