SCHEMBL2597678

SCHEMBL2597678

OB(O)c1cccc(C2CNCCO2)c1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.68
DRD3 P35462 1/20 0.68
HTR1A P08908 1/20 0.59
PRKACA P17612 1/20 0.49
PRKACG P22612 1/20 0.49
PRKACB P22694 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1825157 0.83 DRD2 (0.53) DRD2DRD3
SCHEMBL323312 0.81 DRD3 (1.00) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL2296934 0.81 DRD2 (0.68) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL28215396 0.81 DRD2 (0.68) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL30752418 0.81 DRD2 (0.68) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL2293961 0.81 DRD2 (0.68) DRD2DRD3HTR1APRKACAPRKACG
Hydrochloric Acid SCHEMBL16463508 0.80 DRD2 (0.66) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL16057462 0.80 DRD2 (0.69) DRD2DRD3HTR1APRKACAPRKACG
SCHEMBL28705095 0.78 DRD2 (0.46) DRD2DRD3
SCHEMBL16517709 0.78 DRD2 (0.46) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109890820-B Aminopyrazolopyrimidine compounds as neurotrophin tyrosine kinase receptor inhibitors 正大天晴药业集团股份有限公司 2020-11-03 CN disclosed
CN-111163766-A AHR inhibitors and uses thereof 医肯纳肿瘤学公司 2020-05-15 CN disclosed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
EP-2571856-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed
WO-2011144577-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed