SCHEMBL25985252

SCHEMBL25985252

Brc1ccccc1C1CCOC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.41
HTR2B P41595 4/20 0.41
KDM1A O60341 2/20 0.40
BRD4 O60885 1/20 0.40
SLC6A2 P23975 2/20 0.40
HTR2A P28223 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 1/20 0.40
MAP1LC3B Q9GZQ8 1/20 0.37
BACE1 P56817 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDE10A Q9Y233 2/20 0.34
RCOR1 Q9UKL0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23380370 0.84 HTR2C (0.46) HTR2CHTR2BKDM1ABRD4SLC6A2
SCHEMBL28003145 0.77 KDM1A (0.46) HTR2CHTR2BKDM1ASLC6A2SLC6A4
SCHEMBL28452283 0.77 HTR2C (0.52) HTR2CHTR2BHTR2APDE10A
SCHEMBL29427088 0.77 KDM1A (0.50) HTR2CHTR2BKDM1ABRD4SLC6A2
SCHEMBL10046437 0.77 KDM1A (0.50) HTR2CHTR2BKDM1ABRD4SLC6A2
SCHEMBL23228754 0.74 HTR2C (0.53) HTR2CSLC6A2SLC6A4SLC6A3
SCHEMBL20380077 0.74 CA1 (0.39) CYP2C9F2PLGPLAUPLAT
SCHEMBL21624161 0.73 SLC6A4 (0.55) HTR2CSLC6A4CYP2D6
SCHEMBL1794059 0.73 ALDH1A1 (0.34) ALDH1A1PDE10AF2PLGPLAU
SCHEMBL23662637 0.73 OPRL1 (0.34) SLC6A2SLC6A4SLC6A3ALDH1A1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3814331-B9 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY ORSOBIO INC (US) 2023-08-09 EP disclosed