SCHEMBL2598857

SCHEMBL2598857

CN1CC2c3ccc(CCc4ccccc4)cc3C(=O)NC[C@H]2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
PARP1 P09874 5/20 0.37
NR1H3 Q13133 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
BACE1 P56817 1/20 0.35
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
DPP4 P27487 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ATM Q13315 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
PIM1 P11309 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
PARP3 Q9Y6F1 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861846 1.00 MAOA (0.40) MAOAMAOBPARP1NR1H3TAAR1
SCHEMBL861845 1.00 MAOA (0.40) MAOAMAOBPARP1NR1H3TAAR1
SCHEMBL2598856 1.00 MAOA (0.40) MAOAMAOBPARP1NR1H3TAAR1
SCHEMBL860846 0.83 MEN1 (0.31) S1PR1PIM1PIM2
SCHEMBL860847 0.83 MEN1 (0.31) S1PR1PIM1PIM2
SCHEMBL860696 0.83 MAOA (0.46) MAOAMAOBPARP1S1PR1S1PR5
SCHEMBL2598950 0.83 MAOA (0.46) MAOAMAOBPARP1S1PR1S1PR5
SCHEMBL860697 0.83 MAOA (0.46) MAOAMAOBPARP1S1PR1S1PR5
SCHEMBL861248 0.82 CLK4 (0.44) MAOAMAOBKDM4EHRH3PARP3
SCHEMBL861249 0.82 CLK4 (0.44) MAOAMAOBKDM4EHRH3PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571353-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF AbbVie Inc. (US) 2013-03-27 EP disclosed
WO-2011146089-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-11-24 WO disclosed