SCHEMBL2599342

SCHEMBL2599342

O=C1C(=O)c2cc(Cl)ccc2-c2ccc(Cl)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 5/20 1.00
HSP90AA1 P07900 1/20 0.57
PPOX P50336 1/20 0.56
CES1 P23141 2/20 0.50
TGM2 P21980 1/20 0.50
USP8 P40818 2/20 0.48
USP7 Q93009 2/20 0.48
USP47 Q96K76 1/20 0.48
METAP1 P53582 1/20 0.47
ITGA1 P56199 1/20 0.45
PTPRC P08575 4/20 0.43
MEN1 O00255 1/20 0.43
APAF1 O14727 1/20 0.43
NPC1 O15118 1/20 0.43
TDP2 O95551 1/20 0.43
NSD2 O96028 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
PLA2G1B P04054 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1133148 0.94 S100A4 (0.90) S100A4HSP90AA1PPOXCES1TGM2
SCHEMBL30345128 0.94 S100A4 (0.90) S100A4HSP90AA1PPOXCES1TGM2
SCHEMBL2599398 0.91 S100A4 (1.00) S100A4HSP90AA1PPOXCES1ITGA1
SCHEMBL353693 0.89 S100A4 (0.80) S100A4HSP90AA1PPOXCES1TGM2
SCHEMBL11876117 0.89 S100A4 (0.80) S100A4HSP90AA1PPOXCES1TGM2
SCHEMBL4229683 0.89 S100A4 (0.80) S100A4HSP90AA1PPOXCES1TGM2
SCHEMBL1758264 0.85 S100A4 (0.91) S100A4HSP90AA1PPOXCES1ITGA1
SCHEMBL30419890 0.85 S100A4 (0.91) S100A4HSP90AA1PPOXCES1USP8
SCHEMBL301388 0.85 S100A4 (0.91) S100A4HSP90AA1PPOXCES1USP8
SCHEMBL38651099 0.85 S100A4 (0.91) S100A4HSP90AA1PPOXCES1USP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US claimed
WO-2011146101-A1 CHEMICAL AGENTS FOR THE PREVENTION OR INHIBITION OF TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2011-11-24 WO claimed
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US disclosed
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US disclosed
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-04-11 US disclosed
WO-2011146101-A1 CHEMICAL AGENTS FOR THE PREVENTION OR INHIBITION OF TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2011-11-24 WO disclosed
WO-2011146101-A1 CHEMICAL AGENTS FOR THE PREVENTION OR INHIBITION OF TUMOR METASTASIS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2011-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130090355-A1 CHEMICAL AGENTS FOR THE PREVENTION OF INHIBITION OR TUMOR METASTASIS S100A4, S100A6, S100A10 S100A4 1/4885HSP90AA1 116/4885PPOX 2114/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.