SCHEMBL2599656

SCHEMBL2599656

Fc1cccc2c1OCCN2c1ncc(OCc2ccccc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 3/20 0.40
GRM5 P41594 2/20 0.39
ALKBH1 Q13686 6/20 0.39
MAOB P27338 2/20 0.39
MAOA P21397 1/20 0.39
CYP17A1 P05093 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HTR6 P50406 1/20 0.37
FAAH O00519 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2599617 0.81 PIK3CD (0.43) CYP17A1CYP1A2ALDH1A1HTR6PIK3CD
SCHEMBL2599665 0.77 PIK3CD (0.38) CYP17A1CYP1A2ALDH1A1HTR6PIK3CD
SCHEMBL2599637 0.74 APP (0.41) CYP17A1CYP1A2HTR6PIK3CDPIK3CB
SCHEMBL2599667 0.72 AVPR1A (0.35) CYP17A1CYP1A2HTR6FAAHPIK3CD
SCHEMBL16332713 0.72 CYP17A1 (0.34) CYP17A1CYP1A2HTR6PIK3CDPIK3CB
SCHEMBL16388793 0.71 PIK3CA (0.37) CYP17A1CYP1A2PIK3CDPIK3CBPIK3CG
SCHEMBL28927093 0.69 CYP11B2 (0.62) ALKBH1ALDH1A1KDM4E
SCHEMBL15952657 0.67 KIT (0.54) ALKBH1ALDH1A1
SCHEMBL15953346 0.66 KIT (0.53) ALKBH1ALDH1A1
SCHEMBL26077214 0.66 KIT (0.53) ALKBH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-B1 COMPOUNDS TREHERNE JOHNATHAN MARK (GB) 2014-12-31 EP disclosed
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed