SCHEMBL2599673

SCHEMBL2599673

Fc1cccc2c1OCCN2c1ncc(Oc2cccc(Br)c2)cn1.OC1CN(c2cccc(Oc3cnc(N4CCOc5c(F)cccc54)nc3)c2)C1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.33
DHFR P00374 1/20 0.32
CYP17A1 P05093 1/20 0.32
CYP1A2 P05177 1/20 0.32
PDE4B Q07343 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2599667 0.95 AVPR1A (0.35) AVPR1ADHFRCYP17A1CYP1A2PDE4B
SCHEMBL2599612 0.89 PIK3CD (0.36) AVPR1ACYP17A1CYP1A2PDE4BPIK3CD
SCHEMBL2599623 0.82 DHFR (0.40) DHFRCYP17A1CYP1A2PDE4B
SCHEMBL16332713 0.81 CYP17A1 (0.34) AVPR1ACYP17A1CYP1A2PDE4BPIK3CD
SCHEMBL2599603 0.81 MAPT (0.40) DHFRCYP17A1CYP1A2PIK3CDPIK3CB
SCHEMBL16388603 0.79 F10 (0.37) AVPR1ADHFRCYP17A1CYP1A2PDE4B
SCHEMBL2599613 0.78 DHFR (0.40) DHFRPDE4B
SCHEMBL2599665 0.77 PIK3CD (0.38) AVPR1ADHFRCYP17A1CYP1A2PDE4B
SCHEMBL16388793 0.77 PIK3CA (0.37) AVPR1ACYP17A1CYP1A2PIK3CDPIK3CB
SCHEMBL16332808 0.75 IDH1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571872-A1 COMPOUNDS BTG International Limited (GB) 2013-03-27 EP disclosed
WO-2011144578-A1 COMPOUNDS SENEXIS LIMITED (GB) 2011-11-24 WO disclosed