SCHEMBL2600217

SCHEMBL2600217

CCC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.69
CYP3A4 P08684 1/20 0.67
KCNJ5 P48544 1/20 0.65
KCNJ3 P48549 1/20 0.65
LMNA P02545 5/20 0.64
MAPT P10636 5/20 0.64
ALDH1A1 P00352 3/20 0.64
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
PDK1 Q15118 1/20 0.62
TSHR P16473 1/20 0.61
HTT P42858 1/20 0.60
GAA P10253 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
POLB P06746 1/20 0.57
HPGD P15428 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
TP53 P04637 1/20 0.56
THRB P10828 1/20 0.56
EPHX2 P34913 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26546756 0.89 KDR (0.76) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL29476070 0.87 KDR (0.68) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL2350751 0.87 KDR (0.68) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL13004812 0.86 KDR (0.71) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL4443052 0.86 KDR (0.71) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL27420134 0.86 LMNA (0.63) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL9365319 0.85 KDR (0.66) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL5804247 0.85 KDR (0.69) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL14422910 0.85 KDR (0.69) KDRKCNJ5KCNJ3LMNAMAPT
SCHEMBL28884494 0.85 KDR (0.69) KDRKCNJ5KCNJ3LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109824581-B Alanine-containing peptide-like compound and preparation method and application thereof 西安交通大学 2020-08-18 CN disclosed
CN-109651243-B Serine-containing peptoid compound and preparation method and application thereof 西安交通大学 2020-05-22 CN disclosed
US-8445687-B2 Process for the preparation of a RAF kinase inhibitor and intermediates for use in the process CIPLA LIMITED (IN) 2013-05-21 US disclosed
US-20130029967-A1 Fused Imidazo [3,2 - D] Pyrazines as P13 Kinase Inhibitors CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2013-01-31 US disclosed
US-20120122870-A1 Treatment Of Ischemia-Reperfusion Injury MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2012-05-17 US disclosed
US-20120095004-A1 Sphingosine Kinase Inhibitors APOGEE BIOTECHNOLOGY CORPORATION (US) 2012-04-19 US disclosed
US-8063248-B2 3-(4-Chloro-phenyl)-adamantane-1-carboxylic acidisopropylamide; antiproliferative, antiinflammatory agent, angiogenesis inhibitor; sphingolipid-derived signaling pathway; coupling acid or acylhalide of phenyl-adamantane derivatives with aminoalkyl-pyridine APOGEE BIOTECHNOLOGY CORPORATION (US) 2011-11-22 US disclosed
US-20110046157-A1 Substituted hydroxamic acids and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-02-24 US disclosed
US-20080167352-A1 Sphingosine Kinase Inhibitors APOGEE BIOTECHNOLOGY CORPORATION (US) 2008-07-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130029967-A1 Fused Imidazo [3,2 - D] Pyrazines as P13 Kinase Inhibitors MTOR, PIK3CA, CDK2 KDR 735/4885CYP3A4 902/4885KCNJ5 2301/4885
US-20120095004-A1 Sphingosine Kinase Inhibitors SPHK1, SPHK2, S1PR1 KDR 31/4885CYP3A4 4465/4885KCNJ5 1283/4885
US-20120122870-A1 Treatment Of Ischemia-Reperfusion Injury SPHK1, SPHK2, S1PR2 KDR 719/4885CYP3A4 3146/4885KCNJ5 1584/4885
US-20080167352-A1 Sphingosine Kinase Inhibitors SPHK1, SPHK2, S1PR1 KDR 31/4885CYP3A4 4465/4885KCNJ5 1283/4885
US-20110046157-A1 Substituted hydroxamic acids and uses thereof HDAC6, HDAC5, HDAC1 KDR 2433/4885CYP3A4 3712/4885KCNJ5 3051/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.