SCHEMBL260104

SCHEMBL260104

N#CCc1c[nH]c2cccc([N+](=O)[O-])c12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
HPGD P15428 1/20 0.56
CDK2 P24941 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
BACE1 P56817 2/20 0.43
CSNK2A1 P68400 2/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 2/20 0.41
CLK1 P49759 1/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 2/20 0.40
PKLR P30613 1/20 0.40
RAD52 P43351 1/20 0.39
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL4076350 0.96 ALDH1A1 (0.52) ALDH1A1HPGDCDK2NPC1RAB9A
SCHEMBL12627931 0.81 CDK2 (0.47) ALDH1A1CDK2NPC1RAB9ABACE1
SCHEMBL28770654 0.81 CDK2 (0.46) ALDH1A1CDK2NPC1RAB9ABACE1
SCHEMBL20120186 0.78 HTR2A (0.59) ALDH1A1CDK2NPC1RAB9ABACE1
SCHEMBL259399 0.77 HTR2A (0.58) ALDH1A1CDK2NPC1RAB9ABACE1
SCHEMBL2884596 0.77 ALDH1A1 (0.62) ALDH1A1HPGDCDK2NPC1RAB9A
SCHEMBL261401 0.77 CDK2 (0.44) ALDH1A1CDK2NPC1RAB9ABACE1
SCHEMBL260336 0.77 ALDH1A1 (0.56) ALDH1A1HPGDCDK2NPC1CSNK2A1
SCHEMBL20119875 0.76 KDM4E (0.58) ALDH1A1HPGDCDK2NPC1RAB9A
SCHEMBL2297034 0.76 CLK1 (0.43) ALDH1A1CDK2NPC1RAB9ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573496-B Preparation method of 4-chloroindole-3-acetic acid 贵州大学 2023-11-07 CN disclosed
CN-114573496-A Preparation method of 4-chloroindole-3-acetic acid 贵州大学 2022-06-03 CN disclosed
EP-1951042-B1 SPIROLACTAM TRICYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2012-10-10 EP disclosed
EP-1951051-B1 SPIROHYDANTOIN TRICYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2012-10-03 EP disclosed
US-8163752-B2 Tricyclic anilide heterocyclic CGRP receptor antagonists Merck, Sharp & Dohme Corp. (US) 2012-04-24 US disclosed
US-8133891-B2 Tricyclic anilide spirolactam CGRP receptor antagonists Merck, Sharp & Dohme Corp. (US) 2012-03-13 US disclosed
CN-101076527-B Tricyclic anilide spirohydantoin cgrp receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-11-30 CN disclosed
EP-1794146-B1 TRICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2011-08-03 EP disclosed
US-7968540-B2 Spirohydantoin tricyclic CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-06-28 US disclosed
US-7947677-B2 Spirolactam tricyclic CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-05-24 US disclosed
EP-1951051-A2 SPIROHYDANTOIN TRICYCLIC CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-08-06 EP disclosed
EP-1951042-A2 SPIROLACTAM TRICYCLIC CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-08-06 EP disclosed
CN-101076527-A Tricyclic anilide spirohydantoin cgrp receptor antagonists MERCK & CO INC (US) 2007-11-21 CN disclosed
CN-101014345-A Tricyclic anilide spirolactam cgrp receptor antagonists MERCK & CO INC (US) 2007-08-08 CN disclosed
EP-1793827-A2 TRICYCLIC ANILIDE SPIROLACTAM CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-06-13 EP disclosed
EP-1794146-A2 TRICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-06-13 EP disclosed
WO-2007061694-A2 SPIROHYDANTOIN TRICYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-05-31 WO disclosed
WO-2007061692-A2 SPIROLACTAM TRICYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-05-31 WO disclosed
WO-2006031676-A2 TRICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-03-23 WO disclosed
WO-2006031491-A2 TRICYCLIC ANILIDE SPIROLACTAM CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-03-23 WO disclosed