SCHEMBL26013441

SCHEMBL26013441

Cc1cc(OC(F)(F)F)ccc1CC(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
HRH4 Q9H3N8 2/20 0.40
GPR3 P46089 4/20 0.40
SCN5A Q14524 2/20 0.39
PDE2A O00408 2/20 0.38
CHRM5 P08912 1/20 0.38
CYP1A2 P05177 1/20 0.37
SLC6A4 P31645 1/20 0.37
PSMB5 P28074 1/20 0.37
FFAR4 Q5NUL3 3/20 0.36
SCN10A Q9Y5Y9 3/20 0.36
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36
CACNA1C Q13936 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933301 0.91 SLC6A4 (0.40) PPARGPPARDPPARAHRH4PDE2A
SCHEMBL12414811 0.83 PDE2A (0.48) HRH4GPR3PDE2ACHRM5SLC6A4
SCHEMBL13137672 0.83 GPR3 (0.41) PPARGPPARDPPARAHRH4GPR3
SCHEMBL23998936 0.82 TRPV1 (0.40) PPARDPPARAHRH4GPR3SCN5A
SCHEMBL14143900 0.81 CHRM5 (0.43) PPARGPPARDPPARAGPR3SCN5A
SCHEMBL5018773 0.81 APLNR (0.42)
SCHEMBL17449711 0.80 PDE2A (0.44) HRH4GPR3PDE2ASLC6A4FFAR4
SCHEMBL13568401 0.79 GPR3 (0.41) PPARGPPARDPPARAHRH4GPR3
SCHEMBL20817904 0.79 GPR3 (0.41) PPARGPPARDPPARAHRH4GPR3
SCHEMBL966621 0.79 GPR3 (0.41) PPARGPPARDPPARAHRH4GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154291-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed