SCHEMBL26014646

SCHEMBL26014646

Cc1c(CC(C)C)cccc1OC(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRB2 P47870 1/20 0.43
SLC6A2 P23975 7/20 0.40
SLC6A4 P31645 7/20 0.40
KCNH2 Q12809 5/20 0.37
CYP2D6 P10635 3/20 0.37
SLC6A3 Q01959 4/20 0.37
ESR1 P03372 1/20 0.37
PPARG P37231 2/20 0.36
EPHX2 P34913 1/20 0.36
PDE9A O76083 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
KCNK3 O14649 2/20 0.35
KCNK9 Q9NPC2 2/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2662469 0.84 SLC6A2 (0.49) GABRA1GABRB2SLC6A2SLC6A4KCNH2
SCHEMBL26013438 0.81 GABRA1 (0.42) GABRA1GABRB2SLC6A2SLC6A4SLC6A3
SCHEMBL16956636 0.79 PDCD1 (0.44) SLC6A2SLC6A4SLC6A3KCNK3KCNK9
SCHEMBL13744996 0.79 GABRA1 (0.48) GABRA1GABRB2
SCHEMBL16707610 0.78 HSD11B1 (0.41) SLC6A2SLC6A4SLC6A3KCNK3KCNK9
SCHEMBL22781148 0.75 GABRA1 (0.62) GABRA1GABRB2SLC6A2SLC6A4KCNH2
SCHEMBL21283351 0.74 GABRA1 (0.52) GABRA1GABRB2SLC6A2SLC6A4KCNH2
SCHEMBL20847853 0.74 KCNK3 (0.49) KCNK3KCNK9
SCHEMBL16159968 0.74 KCNK3 (0.49) GABRA1GABRB2SLC6A2KCNK3KCNK9
SCHEMBL17449715 0.73 KCNH2 (0.41) SLC6A2SLC6A4KCNH2CYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154291-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed