SCHEMBL2601907

SCHEMBL2601907

CC(C)n1c(=O)oc2cc(NC(=O)N[C@H]3CC[C@H](NS(=O)(=O)C(C)(C)C)CC3)ccc21

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
EPHX2 P34913 4/20 0.38
GNRHR P30968 1/20 0.38
POLB P06746 1/20 0.37
MMP12 P39900 1/20 0.37
MMP13 P45452 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPT P10636 1/20 0.37
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2601694 0.89 NPY5R (0.41) ALDH1A1EPHX2GNRHRPOLBMMP12
SCHEMBL2601692 0.88 TP53 (0.40) ALDH1A1EPHX2GNRHRMAPT
SCHEMBL2600317 0.86 NPY5R (0.41) ALDH1A1MAPTLMNAHPGDTSHR
SCHEMBL11936157 0.83 ALDH1A1 (0.37) ALDH1A1MAPTLMNAHPGDTSHR
SCHEMBL2600321 0.82 EPHX2 (0.56) ALDH1A1EPHX2CYP2C19
SCHEMBL2601891 0.79 KDM4E (0.41) ALDH1A1POLBMAPTTSHR
SCHEMBL2600311 0.76 NPY5R (0.43) ALDH1A1MAPTLMNAHPGDTSHR
SCHEMBL11936280 0.76 NPY5R (0.37) ALDH1A1LMNAHPGDTSHR
SCHEMBL2600316 0.75 NPY5R (0.43) ALDH1A1MAPTLMNAHPGDTSHR
SCHEMBL2600313 0.74 ALDH1A1 (0.46) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8372833-B2 Urea derivative SHIONOGI & CO., LTD. (JP) 2013-02-12 US disclosed
US-20120095231-A1 UREA DERIVATIVE YANO TOSHISADA (JP) 2012-04-19 US disclosed
US-8088777-B2 Urea derivative SHIONOGI & CO., LTD. (JP) 2012-01-03 US disclosed
US-8088777-B2 Urea derivative SHIONOGI & CO., LTD. (JP) 2012-01-03 US disclosed
US-20090203712-A1 Urea Derivative SHIONOGI &CO., LTD. 2009-08-13 US disclosed
US-20090203712-A1 Urea Derivative SHIONOGI &CO., LTD. 2009-08-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095231-A1 UREA DERIVATIVE NPY5R, NPY1R, NPY2R ALDH1A1 4384/4885EPHX2 4211/4885GNRHR 83/4885
US-20090203712-A1 Urea Derivative NPY5R, NPY1R, NPY2R ALDH1A1 4390/4885EPHX2 4206/4885GNRHR 80/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.