SCHEMBL26026993

SCHEMBL26026993

Cc1cccc2c(Oc3c(Cl)cc(N)cc3Cl)n[nH]c(=O)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARG P13631 3/20 0.44
PARP1 P09874 3/20 0.37
LMNA P02545 2/20 0.36
TSHR P16473 1/20 0.36
TNKS O95271 2/20 0.35
TNKS2 Q9H2K2 2/20 0.35
AR P10275 4/20 0.34
CHEK1 O14757 2/20 0.34
RORC P51449 2/20 0.34
TYMS P04818 2/20 0.33
DRD1 P21728 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
FLT3 P36888 1/20 0.32
PLK3 Q9H4B4 1/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
CYP2C9 P11712 1/20 0.32
UGT1A1 P22309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26026689 0.89 RARG (0.50) RARGPARP1LMNAARCHEK1
SCHEMBL26027584 0.86 RARG (0.42) RARGPARP1LMNATSHRTNKS
SCHEMBL26026865 0.86 RARG (0.44) RARGPARP1LMNAARCHEK1
SCHEMBL22077248 0.82 RARG (0.50) RARGPARP1LMNATSHRAR
SCHEMBL29578026 0.82 RARG (0.50) RARGPARP1LMNATSHRAR
SCHEMBL24375457 0.77 THRB (0.36) RARGLMNATSHRDRD1THRA
SCHEMBL26027125 0.77 RARG (0.39) RARGLMNAARTYMSHTT
SCHEMBL22108436 0.76 THRA (0.58) THRATHRBCYP2C9UGT1A1ABCG2
SCHEMBL25430197 0.76 GAA (0.42) RARGPARP1DRD1PARP2THRA
SCHEMBL26027437 0.75 RARG (0.33) RARGPARP1THRATHRBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154842-A1 THR BETA ANALOGS AND USES THEREOF MADRIGAL PHARMACEUTICALS, INC. (US) 2023-08-17 WO disclosed