SCHEMBL26039613

SCHEMBL26039613

CNC(=O)c1cc(OCC(F)F)nn1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.39
PKM P14618 1/20 0.38
BAZ2B Q9UIF8 1/20 0.38
GABRA5 P31644 4/20 0.36
BRD4 O60885 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NTRK1 P04629 1/20 0.35
NTRK3 Q16288 1/20 0.35
JMJD6 Q6NYC1 1/20 0.35
SCN9A Q15858 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HIF1A Q16665 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25349897 0.84 KDM4E (0.44) PKMGABRA5JMJD6SCN9AALDH1A1
SCHEMBL25999611 0.80 CCNE1 (0.40) PKMGABRA5L3MBTL1MEN1KMT2A
SCHEMBL17517052 0.72 BAZ2B (0.41) BAZ2BBRD4L3MBTL1MEN1KMT2A
SCHEMBL24799262 0.72 BAZ2B (0.51) BAZ2BBRD4L3MBTL1MEN1KMT2A
SCHEMBL27239565 0.72 CDK2 (0.45)
SCHEMBL17473215 0.71 PKM (0.37) PKMBAZ2BBRD4L3MBTL1ALDH1A1
SCHEMBL31667472 0.70 CA12 (0.39) PKMGABRA5L3MBTL1JMJD6MEN1
SCHEMBL2737317 0.69 BAZ2B (0.46) BAZ2BBRD4L3MBTL1MEN1KMT2A
SCHEMBL8568508 0.69 SMN1; SMN2 (0.56) BAZ2BL3MBTL1NTRK1MEN1KMT2A
SCHEMBL27258704 0.69 JMJD6 (0.32) PKMJMJD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154426-A1 CDK INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed