SCHEMBL26046397

SCHEMBL26046397

COc1ccc(/C=C/C(C)=O)c(CO)c1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
FDPS P14324 1/20 0.46
APP P05067 5/20 0.46
BACE1 P56817 3/20 0.44
IAPP P10997 1/20 0.43
ABCB1 P08183 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
NFE2L2 Q16236 1/20 0.41
TLR2 O60603 1/20 0.41
ERN1 O75460 1/20 0.41
TLR1 Q15399 1/20 0.41
TLR6 Q9Y2C9 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
JUN P05412 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26046331 0.88 PKM (0.49) KDM4EAPPBACE1GAAMAPT
SCHEMBL26046395 0.85 KDM4E (0.53) KDM4EFDPSAPPBACE1ABCB1
SCHEMBL26046382 0.83 KDM4E (0.60) KDM4EFDPSAPPBACE1IAPP
SCHEMBL26046384 0.81 IAPP (0.56) KDM4EAPPIAPPMAPTLMNA
SCHEMBL26046486 0.81 CYP3A4 (0.42) KDM4EAPPBACE1MAPTLMNA
SCHEMBL26046367 0.81 KDM4E (0.67) KDM4EFDPSBACE1IAPPMAPT
SCHEMBL1877093 0.80 KDM4E (0.57) KDM4EFDPSAPPIAPPABCB1
SCHEMBL1877092 0.80 KDM4E (0.57) KDM4EFDPSAPPIAPPABCB1
SCHEMBL26046381 0.79 APP (0.46) KDM4EAPPBACE1IAPPABCB1
SCHEMBL26046380 0.77 KDM4E (0.57) KDM4EFDPSAPPIAPPABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11746364-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-09-05 US disclosed
US-11739354-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-08-29 US disclosed