SCHEMBL26057778

SCHEMBL26057778

C[C@H]1C[C@@]2(CCN1)OCCc1sccc12

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.46
KCNH2 Q12809 3/20 0.40
DRD3 P35462 1/20 0.34
GID4 Q8IVV7 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
KEAP1 Q14145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25358161 1.00 SIGMAR1 (0.46) SIGMAR1KCNH2DRD3GID4TAAR1
SCHEMBL25355241 0.82 TAAR1 (0.42) SIGMAR1TAAR1
SCHEMBL25357922 0.82 TAAR1 (0.42) SIGMAR1TAAR1
SCHEMBL25358590 0.82 TAAR1 (0.42) SIGMAR1TAAR1
SCHEMBL14906788 0.79 SIGMAR1 (0.56) SIGMAR1KCNH2TAAR1
SCHEMBL25355547 0.78 PNMT (0.32)
SCHEMBL25357944 0.78 PNMT (0.32)
SCHEMBL31387328 0.78 PNMT (0.32)
SCHEMBL25358449 0.78 PNMT (0.32)
SCHEMBL25357162 0.78 PNMT (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154344-A1 2-METHYL-4',5'-DIHYDROSPIRO[PIPERIDINE-4,7'-THIENO[2,3-C]PYRAN] DERIVATIVES AS INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed