SCHEMBL2605799

SCHEMBL2605799

O=[N+]([O-])c1ccc(-c2nc3ccccc3n2-c2ccccc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.72
HTT P42858 3/20 0.72
RXFP1 Q9HBX9 2/20 0.67
PKM P14618 1/20 0.67
RAB9A P51151 1/20 0.67
POLB P06746 1/20 0.59
ESR1 P03372 1/20 0.56
ESR2 Q92731 1/20 0.56
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
KDM4E B2RXH2 1/20 0.55
PTGS2 P35354 1/20 0.52
MAOA P21397 1/20 0.52
GRIA1 P42261 1/20 0.51
CACNG8 Q8WXS5 1/20 0.51
CACNG2 Q9Y698 1/20 0.51
CFTR P13569 1/20 0.50
RECQL P46063 1/20 0.49
MAPK1 P28482 1/20 0.49
ADORA2A P29274 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28142999 0.94 ALDH1A1 (0.64) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL2602407 0.91 ALDH1A1 (0.72) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL28283489 0.89 ALDH1A1 (0.65) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL28142270 0.85 ALDH1A1 (0.56) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL8025343 0.85 HTT (0.58) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL804992 0.85 ESR2 (0.73) ALDH1A1HTTPKMRAB9AESR1
SCHEMBL2326368 0.85 ALDH1A1 (0.63) ALDH1A1HTTRXFP1PKMRAB9A
SCHEMBL10041513 0.83 ESR2 (0.71) ALDH1A1HTTPKMRAB9AESR1
SCHEMBL16692234 0.83 ESR2 (0.71) ALDH1A1HTTPKMRAB9AESR1
SCHEMBL23336889 0.83 ALDH1A1 (0.66) ALDH1A1HTTRXFP1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210130382-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT EMITTING DIODE AND ORGANIC LIGHT EMITTING DEVICE INCLUDING THE SAME LG DISPLAY CO., LTD. (KR) 2021-05-06 US disclosed
CN-104557725-B A kind of method of the diaryl benzimidazole of one pot process 1,2 and its derivative 江苏先科药业有限公司 2017-06-30 CN disclosed
US-8362019-B2 Synthesis and anti-proliferative effect of substituted imidazo[4,5-b]pyrazine compounds SPELMAN COLLEGE (US) 2013-01-29 US disclosed
US-20120095009-A1 SYNTHESIS AND ANTI-PROLIFERATIVE EFFECT OF BENZIMIDAZOLE DERIVATIVES SPELMAN COLLEGE (US) 2012-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210130382-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT EMITTING DIODE AND ORGANIC LIGHT EMITTING DEVICE INCLUDING THE SAME DDT, ORC3, PPOX ALDH1A1 195/4885HTT 3669/4885RXFP1 4815/4885
US-20120095009-A1 SYNTHESIS AND ANTI-PROLIFERATIVE EFFECT OF BENZIMIDAZOLE DERIVATIVES MKI67, CCNI, TYMP ALDH1A1 1026/4885HTT 4534/4885RXFP1 4777/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.