SCHEMBL26066566

SCHEMBL26066566

COc1cc2ccnc(Nc3ccc(F)c(C)c3)c2cc1C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 5/20 0.60
GRM4 Q14833 2/20 0.46
EGFR P00533 7/20 0.44
KDR P35968 3/20 0.44
FBP1 P09467 2/20 0.44
ERBB2 P04626 2/20 0.44
RET P07949 2/20 0.44
KIF5B P33176 2/20 0.44
AURKA O14965 1/20 0.44
INSR P06213 1/20 0.44
PDGFRB P09619 1/20 0.44
FLT4 P35916 1/20 0.44
CLK1 P49759 1/20 0.44
EPHB4 P54760 1/20 0.44
TEK Q02763 1/20 0.44
AURKB Q96GD4 1/20 0.44
RIPK2 O43353 1/20 0.44
NOD1 Q9Y239 1/20 0.44
PIK3CA P42336 2/20 0.43
TRPA1 O75762 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26066568 0.90 TNF (0.63) TNFEGFRKDRFBP1ERBB2
SCHEMBL26066602 0.89 TNF (0.61) TNFEGFRKDRERBB2RET
SCHEMBL26066662 0.88 TNF (0.49) TNFGRM4EGFRFBP1ERBB2
SCHEMBL26066665 0.87 GRM4 (0.48) TNFGRM4EGFRKDRPIK3CA
SCHEMBL26066664 0.87 TNF (0.48) TNFGRM4EGFRKDRFBP1
SCHEMBL26066599 0.83 TNF (0.64) TNFGRM4EPHB4
SCHEMBL26066601 0.82 TNF (0.50) TNFGRM4EGFRKDRFBP1
SCHEMBL26066598 0.82 TNF (0.57) TNFGRM4EGFRKDRFBP1
SCHEMBL26066603 0.81 TNF (0.45) TNFGRM4EGFRKDRFBP1
SCHEMBL23624399 0.80 TNF (0.62) TNFEGFRCLK1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023155019-A1 ISOQUINOLINE DERIVATIVES AS INHIBITORS OF BAX AND/OR BAK, COMPOSITIONS AND USES THEREOF Sunnybrook Research Institute (CA) 2023-08-24 WO disclosed