SCHEMBL26089322

SCHEMBL26089322

CCOC(=O)c1ccc(C)c(C2CCN(Cc3ccccc3)C2)c1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRMT1 Q99873 1/20 0.54
MAPK1 P28482 1/20 0.50
LMNA P02545 1/20 0.50
DRD2 P14416 2/20 0.48
DRD4 P21917 2/20 0.48
TSHR P16473 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.46
CCR8 P51685 1/20 0.45
SCN4A P35499 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31313650 1.00 PRMT1 (0.54) PRMT1MAPK1LMNADRD2DRD4
SCHEMBL27042396 0.90 KDM4E (0.47) PRMT1MAPK1LMNATSHRALDH1A1
SCHEMBL27042601 0.88 DRD4 (0.50) LMNADRD2DRD4SCN4A
SCHEMBL26092030 0.82 FDFT1 (0.46) MAPK1ALDH1A1KDM4E
SCHEMBL26093038 0.82 FDFT1 (0.46) MAPK1ALDH1A1KDM4E
SCHEMBL27042490 0.81 PRMT1 (0.50) PRMT1MAPK1LMNATSHRALDH1A1
SCHEMBL30728773 0.81 PRMT1 (0.50) PRMT1MAPK1LMNATSHRALDH1A1
SCHEMBL30728803 0.81 PRMT1 (0.50) PRMT1MAPK1LMNATSHRALDH1A1
SCHEMBL31533977 0.80 TSHR (0.50) PRMT1DRD2DRD4TSHRALDH1A1
SCHEMBL30728753 0.80 PRMT1 (0.49) PRMT1MAPK1LMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4558489-A1 HETEROARYL DERIVATIVES AS DDRs INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2025-05-28 EP disclosed
EP-4419516-A1 PYRROLIDINE DERIVATIVES AS DDRS INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2024-08-28 EP disclosed
CN-118284601-A Pyrrolidine derivatives as DDR inhibitors 奇斯药制品公司 2024-07-02 CN disclosed
WO-2024017876-A1 HETEROARYL DERIVATIVES AS DDRs INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2024-01-25 WO disclosed
WO-2024017876-A1 HETEROARYL DERIVATIVES AS DDRs INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2024-01-25 WO disclosed
WO-2023066834-A1 PYRROLIDINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-04-27 WO disclosed
WO-2023066834-A1 PYRROLIDINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-04-27 WO disclosed