SCHEMBL261010

SCHEMBL261010

Nc1ccc(Nc2c(Nc3ccc(N)cc3)c(=O)c2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
ALOX12 P18054 1/20 0.52
CYP2C19 P33261 1/20 0.52
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
RAD52 P43351 1/20 0.48
KDM1A O60341 1/20 0.47
CXCR2 P25025 4/20 0.46
NR4A1 P22736 1/20 0.45
KDM4E B2RXH2 1/20 0.45
TP53 P04637 1/20 0.45
APP P05067 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
SNCA P37840 1/20 0.45
BLM P54132 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL8359601 0.98 MAPT (0.50) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL5438258 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL12747008 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL18289620 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL5428343 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL29479572 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL33864 0.78 MAPT (0.78) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL1459001 0.75 MAPT (0.74) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL8440919 0.75 MAPT (0.74) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL24137170 0.75 CXCR2 (0.66) MAPTALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071282-B2 Benzimidazole diamine-based polyetherimide compositions and methods for making them GENERAL ELECTRIC COMPANY (US) 2006-07-04 US claimed
EP-1633802-A1 BENZIMIDAZOLE DIAMINE-BASED POLYETHERIMIDE COMPOSITIONS AND METHODS FOR MAKING THEM GENERAL ELECTRIC COMPANY (US) 2006-03-15 EP claimed
WO-2004108797-A1 BENZIMIDAZOLE DIAMINE-BASED POLYETHERIMIDE COMPOSITIONS AND METHODS FOR MAKING THEM GENERAL ELECTRIC COMPANY (US) 2004-12-16 WO claimed
US-20040249117-A1 Benzimidazole diamine-based polyetherimide compositions and methods for making them GENERAL ELECTRIC COMPANY 2004-12-09 US claimed
US-5889139-A PREPARED USING EQUIMOLAR AMOUNT OF DIANHYDRIDE AND COMBINATION OF DIAMINES; ENCAPSULANTS, INTERLAYER DIELECTRICS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1999-03-30 US claimed
US-5212283-A Films and adhesives THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1993-05-18 US claimed
EP-2280963-B1 METHOD OF PURIFYING DIANHYDRIDES, THE DIANHYDRIDES FORMED THEREBY, AND POLYETHERIMIDES FORMED THEREFROM SABIC GLOBAL TECHNOLOGIES BV (NL) 2016-07-20 EP disclosed
EP-2097375-B1 METHOD FOR PURIFYING BISIMIDES SABIC INNOVATIVE PLASTICS IP (NL) 2013-04-24 EP disclosed
EP-2089348-B1 METHOD FOR MAKING POLYETHERIMIDES SABIC INNOVATIVE PLASTICS IP (NL) 2013-02-20 EP disclosed
US-8134016-B2 Method for purifying dianhydrides SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2012-03-13 US disclosed
US-8013173-B2 Method of purifying dianhydrides, the dianhydrides formed thereby, and polyetherimides formed therefrom SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2011-09-06 US disclosed
EP-2094691-B1 METHOD FOR PURIFYING DIANHYDRIDES SABIC INNOVATIVE PLASTICS IP (NL) 2011-05-25 EP disclosed
EP-2280963-A1 METHOD OF PURIFYING DIANHYDRIDES, THE DIANHYDRIDES FORMED THEREBY, AND POLYETHERIMIDES FORMED THEREFROM SABIC Innovative Plastics IP B.V. (NL) 2011-02-09 EP disclosed
US-7071282-B2 Benzimidazole diamine-based polyetherimide compositions and methods for making them GENERAL ELECTRIC COMPANY (US) 2006-07-04 US disclosed
US-20040265605-A1 Data storage medium comprising polyimides GENERAL ELECTRIC COMPANY 2004-12-30 US disclosed
US-20040249117-A1 Benzimidazole diamine-based polyetherimide compositions and methods for making them GENERAL ELECTRIC COMPANY 2004-12-09 US disclosed
US-5889139-A PREPARED USING EQUIMOLAR AMOUNT OF DIANHYDRIDE AND COMBINATION OF DIAMINES; ENCAPSULANTS, INTERLAYER DIELECTRICS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1999-03-30 US disclosed
EP-0558894-B1 Squaric acid derivatives KYOWA HAKKO KOGYO KK (JP) 1996-05-01 EP disclosed
US-5212283-A Films and adhesives THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1993-05-18 US disclosed
US-5212283-A Films and adhesives THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1993-05-18 US disclosed