SCHEMBL26102488

SCHEMBL26102488

CC(=O)OC[C@H]1OC(O)[C@H](OC(C)=O)[C@@H](OCc2ccc3ccccc3c2)[C@@H]1OC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
PYGL P06737 1/20 0.49
POLB P06746 1/20 0.48
LMNA P02545 3/20 0.45
SSTR4 P31391 2/20 0.44
SSTR1 P30872 1/20 0.44
SSTR2 P30874 1/20 0.44
SSTR3 P32745 1/20 0.44
SSTR5 P35346 1/20 0.44
CA12 O43570 6/20 0.43
CA9 Q16790 6/20 0.43
CA1 P00915 5/20 0.43
CA2 P00918 4/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA5A P35218 2/20 0.43
CA7 P43166 2/20 0.43
CA13 Q8N1Q1 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA5B Q9Y2D0 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19457698 0.90 POLB (0.53) TSHRPYGLPOLBLMNASSTR4
SCHEMBL30612814 0.90 POLB (0.53) TSHRPYGLPOLBLMNASSTR4
SCHEMBL21219187 0.87 TSHR (0.59) TSHRPOLBLMNACA12CA9
SCHEMBL17502058 0.87 TSHR (0.59) TSHRPOLBLMNACA12CA9
SCHEMBL19457702 0.85 KDM4E (0.47) TSHRPYGLPOLBLMNASSTR4
SCHEMBL17502089 0.82 TSHR (0.62) TSHRPOLBLMNACA12CA9
SCHEMBL17502004 0.82 TSHR (0.59) TSHRPOLBLMNACA12CA9
SCHEMBL26517127 0.82 POLB (0.47) TSHRPYGLPOLBLMNASSTR4
SCHEMBL13380996 0.79 TSHR (0.50) TSHRPOLBLMNASSTR4SSTR1
SCHEMBL20287904 0.79 TSHR (0.50) TSHRPOLBLMNASSTR4SSTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250346622-A1 NOVEL OLIGOSACCHARIDE, MANUFACTURING INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, AND METHOD FOR MANUFACTURING THESE DAIICHI SANKYO COMPANY, LIMITED (JP) 2025-11-13 US disclosed
EP-4585601-A1 NOVEL OLIGOSACCHARIDE, PRODUCTION INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, PRODUCTION METHOD FOR NOVEL OLIGOSACCHARIDE, AND PRODUCTION METHOD FOR PRODUCTION INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE Daiichi Sankyo Company, Limited (JP) 2025-07-16 EP disclosed
EP-4424717-A1 NOVEL OLIGOSACCHARIDE, MANUFACTURING INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, AND METHOD FOR MANUFACTURING THESE Daiichi Sankyo Company, Limited (JP) 2024-09-04 EP disclosed
US-20240279364-A1 GLYCAN, AND METHOD FOR PRODUCING MEDICINE CONTAINING GLYCAN DAIICHI SANKYO COMPANY, LIMITED (JP) 2024-08-22 US disclosed
CN-118302451-A Novel oligosaccharide, intermediate for producing the oligosaccharide, and process for producing the same 第一三共株式会社 2024-07-05 CN disclosed
WO-2024053574-A1 NOVEL OLIGOSACCHARIDE, PRODUCTION INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, PRODUCTION METHOD FOR NOVEL OLIGOSACCHARIDE, AND PRODUCTION METHOD FOR PRODUCTION INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE 第一三共株式会社 2024-03-14 WO disclosed
EP-4306546-A1 GLYCAN, AND METHOD FOR PRODUCING MEDICINE CONTAINING GLYCAN Daiichi Sankyo Company, Limited (JP) 2024-01-17 EP disclosed
CN-116917341-A Sugar chain and method for producing pharmaceutical product containing sugar chain 第一三共株式会社 2023-10-20 CN disclosed
WO-2023074843-A1 NOVEL OLIGOSACCHARIDE, MANUFACTURING INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, AND METHOD FOR MANUFACTURING THESE 第一三共株式会社 2023-05-04 WO disclosed
WO-2022191313-A1 GLYCAN, AND METHOD FOR PRODUCING MEDICINE CONTAINING GLYCAN 第一三共株式会社 2022-09-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240279364-A1 GLYCAN, AND METHOD FOR PRODUCING MEDICINE CONTAINING GLYCAN FUT6, ST6GAL1, NEU2 TSHR 1157/4885PYGL 462/4885POLB 4077/4885
US-20250346622-A1 NOVEL OLIGOSACCHARIDE, MANUFACTURING INTERMEDIATE FOR NOVEL OLIGOSACCHARIDE, AND METHOD FOR MANUFACTURING THESE FUT6, FUT5, ST3GAL3 TSHR 2600/4885PYGL 2278/4885POLB 4505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.