SCHEMBL26114657

SCHEMBL26114657

COc1cc(F)ccc1-c1nnc(N[C@@H]2C[C@@H](F)CN(C(=O)O)C2)c2ccncc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 10/20 0.37
CASP3 P42574 3/20 0.37
CASP7 P55210 3/20 0.37
KDM4C Q9H3R0 1/20 0.36
CCNT1 O60563 6/20 0.35
PIP4K2A P48426 1/20 0.35
KCNH2 Q12809 3/20 0.35
GRIN2B Q13224 1/20 0.35
BTK Q06187 1/20 0.34
CDK1 P06493 2/20 0.34
CDK2 P24941 2/20 0.34
CDK3 Q00526 2/20 0.34
CDK5 Q00535 2/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNE1 P24864 1/20 0.34
CCNA1 P78396 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26118444 0.97 CDK9 (0.37) CDK9CASP3CASP7KDM4CCCNT1
SCHEMBL26515018 0.90 GPBAR1 (0.45) CDK9CCNT1
SCHEMBL31359746 0.90 GPBAR1 (0.45) CDK9CCNT1
SCHEMBL26115214 0.87 CDK9 (0.38) CDK9CASP3CASP7CCNT1KCNH2
SCHEMBL31359797 0.87 CDK9 (0.38) CDK9CASP3CASP7CCNT1KCNH2
SCHEMBL26515016 0.87 GPBAR1 (0.45) CDK9CCNT1
SCHEMBL31359734 0.87 GPBAR1 (0.45) CDK9CCNT1
SCHEMBL31359756 0.84 CCNT1 (0.38) CDK9CASP3CASP7CCNT1KCNH2
SCHEMBL26113292 0.84 CCNT1 (0.38) CDK9CASP3CASP7CCNT1KCNH2
SCHEMBL26120739 0.84 EGFR (0.37) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023194964-A1 FUSED PYRIDAZINE DERIVATIVES AS NLRP3 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-12 WO disclosed