SCHEMBL26515016

SCHEMBL26515016

COc1cc(F)ccc1-c1nnc(N[C@@H]2C[C@@H](F)CN(C(=O)OC(C)(C)C)C2)c2cnccc12

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.45
CCNT1 O60563 9/20 0.41
CDK9 P50750 9/20 0.41
DNMT3A Q9Y6K1 1/20 0.41
NSD2 O96028 1/20 0.38
PIK3CD O00329 2/20 0.37
EHMT2 Q96KQ7 1/20 0.37
PDE4B Q07343 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31359734 1.00 GPBAR1 (0.45) GPBAR1CCNT1CDK9DNMT3ANSD2
SCHEMBL31359746 0.97 GPBAR1 (0.45) GPBAR1CCNT1CDK9DNMT3ANSD2
SCHEMBL26515018 0.97 GPBAR1 (0.45) GPBAR1CCNT1CDK9DNMT3ANSD2
SCHEMBL26118444 0.90 CDK9 (0.37) CCNT1CDK9
SCHEMBL26515040 0.88 DYRK1A (0.41) GPBAR1DNMT3ANSD2PIK3CD
SCHEMBL31359830 0.88 DYRK1A (0.41) GPBAR1DNMT3ANSD2PIK3CD
SCHEMBL26114657 0.87 CDK9 (0.37) CCNT1CDK9
SCHEMBL31359866 0.85 CYP3A4 (0.42) MKNK1
SCHEMBL26515093 0.85 CYP3A4 (0.42) MKNK1
SCHEMBL31359756 0.84 CCNT1 (0.38) CCNT1CDK9EHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023194964-A1 FUSED PYRIDAZINE DERIVATIVES AS NLRP3 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-12 WO disclosed