SCHEMBL261247

SCHEMBL261247

CC(C)(C)[Si](OC[C@@H]1C[C@@H]2C[C@@]2(Cc2ccccc2)CN1C(=O)O)(c1ccccc1)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 3/20 0.34
ALDH1A1 P00352 3/20 0.33
HPGD P15428 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
OPRK1 P41145 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387131 0.83 SMYD2 (0.36) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL31298376 0.79 SMYD2 (0.38) SMYD2ALDH1A1HPGDCYP3A4HTT
SCHEMBL31298390 0.77 SMYD2 (0.41) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL263781 0.77 ALDH1A1 (0.39) ALDH1A1HPGDOPRK1HSD11B1
SCHEMBL25364479 0.76 RIPK1 (0.42) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL18587707 0.76 RIPK1 (0.42) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL25365732 0.76 RIPK1 (0.42) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL2146189 0.76 RIPK1 (0.42) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL18587235 0.75 SMYD2 (0.36) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL2795827 0.75 SMYD2 (0.36) SMYD2ALDH1A1CYP3A4HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133908-B2 Heteroaryl derivatives of N-{[(1S,4S,6S)-3-(2-pyridinylcarbonyl)-3-azabicyclo[4.1.0]hept-4-yl]methyl}-2-amine GLAXO GROUP LIMITED (GB) 2012-03-13 US disclosed