SCHEMBL2615364

SCHEMBL2615364

CN1CCN(C2=Nc3cc([18F])ccc3Nc3ccccc32)CC1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 8/20 0.84
HRH1 P35367 2/20 0.84
PAK1 Q13153 1/20 0.84
DRD2 P14416 3/20 0.74
DRD4 P21917 3/20 0.74
DRD3 P35462 2/20 0.74
MAPK1 P28482 2/20 0.74
HTR3E A5X5Y0 1/20 0.74
MEN1 O00255 1/20 0.74
CACNA1F O60840 1/20 0.74
HTR3B O95264 1/20 0.74
ABCB11 O95342 1/20 0.74
LMNA P02545 1/20 0.74
CYP1A2 P05177 1/20 0.74
POLB P06746 1/20 0.74
ADRB2 P07550 1/20 0.74
CHRM2 P08172 1/20 0.74
CHRM4 P08173 1/20 0.74
CYP3A4 P08684 1/20 0.74
HTR1A P08908 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2615365 1.00 CHRM1 (0.84) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL21258026 0.88 CHRM1 (0.65) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL9013860 0.86 CHRM1 (1.00) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL3414200 0.86 CHRM1 (0.74) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL21234807 0.86 CHRM1 (0.78) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL7410410 0.86 CHRM1 (0.73) CHRM1HRH1PAK1DRD2DRD4
SCHEMBL141020 0.86 DRD2 (1.00) CHRM1HRH1DRD2DRD4DRD3
SCHEMBL29470861 0.86 DRD2 (1.00) CHRM1HRH1DRD2DRD4DRD3
Clozapine SCHEMBL20876213 0.85 DRD2 (1.00) CHRM1HRH1DRD2DRD4DRD3
Clozapine SCHEMBL5501558 0.85 DRD2 (1.00) CHRM1HRH1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120095217-A1 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2012-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095217-A1 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF FLI1, CDC73, FOS CHRM1 4388/4885HRH1 4629/4885PAK1 964/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.