SCHEMBL2623698

SCHEMBL2623698

CCOC(=O)CCc1ccc(OC)c(C(=O)CCCCN2C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
LMNA P02545 1/20 0.49
GAA P10253 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
TSHR P16473 2/20 0.47
MAPK1 P28482 2/20 0.47
GLA P06280 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
HTT P42858 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2623700 0.85 ALDH1A1 (0.57) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL4458645 0.82 CYP3A4 (0.50) ALDH1A1GAAL3MBTL1CYP3A4CYP2C9
SCHEMBL9798967 0.79 ALDH1A1 (0.58) ALDH1A1LMNAL3MBTL1CYP3A4CYP2C9
SCHEMBL9798508 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL7547276 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL7549194 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL7543946 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL2618100 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL7589770 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4
SCHEMBL7543605 0.77 HDAC8 (0.59) ALDH1A1LMNAGAAL3MBTL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8772226-B2 Methods and compositions for the detection of cancer THE JOHNS HOPKINS UNIVERSITY (US) 2014-07-08 US disclosed
US-8772226-B2 Methods and compositions for the detection of cancer THE JOHNS HOPKINS UNIVERSITY (US) 2014-07-08 US disclosed
US-20120093724-A1 METHODS AND COMPOSITIONS FOR THE DETECTION OF CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2012-04-19 US disclosed
US-20120093724-A1 METHODS AND COMPOSITIONS FOR THE DETECTION OF CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2012-04-19 US disclosed
WO-2010107909-A2 METHODS AND COMPOSITIONS FOR THE DETECTION OF CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2010-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120093724-A1 METHODS AND COMPOSITIONS FOR THE DETECTION OF CANCER KLK3, KLK2, KLK5 ALDH1A1 1673/4885LMNA 1949/4885GAA 367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.