SCHEMBL2626536

SCHEMBL2626536

O=C1C[C@@H](N2CCCc3ccccc32)C(=O)N1c1ccc(S(=O)(=O)Nc2nccs2)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
GAA P10253 5/20 0.51
GFER P55789 3/20 0.51
KMT2A Q03164 4/20 0.51
SCN9A Q15858 7/20 0.51
MAPT P10636 3/20 0.48
MEN1 O00255 2/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 2/20 0.44
USP2 O75604 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MCL1 Q07820 1/20 0.43
SCN1B Q07699 1/20 0.42
SCN8A Q9UQD0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2626701 1.00 ALDH1A1 (0.59) ALDH1A1GAAGFERKMT2ASCN9A
SCHEMBL10310857 1.00 ALDH1A1 (0.59) ALDH1A1GAAGFERKMT2ASCN9A
SCHEMBL1576404 0.89 KMT2A (0.48) ALDH1A1KMT2ASCN9ALMNASCN1B
SCHEMBL12709026 0.89 KMT2A (0.48) ALDH1A1KMT2ASCN9ALMNASCN1B
SCHEMBL2626698 0.89 KMT2A (0.48) ALDH1A1KMT2ASCN9ALMNASCN1B
SCHEMBL2625918 0.86 SCN9A (0.52) ALDH1A1KMT2ASCN9AMEN1LMNA
SCHEMBL2626679 0.86 SCN9A (0.52) ALDH1A1KMT2ASCN9AMEN1LMNA
SCHEMBL2626065 0.81 KMT2A (0.52) ALDH1A1KMT2ASCN9AMEN1LMNA
SCHEMBL1576529 0.81 KMT2A (0.52) ALDH1A1KMT2ASCN9AMEN1LMNA
SCHEMBL1576703 0.81 KMT2A (0.52) ALDH1A1KMT2ASCN9AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163720-B2 Pyrrolidinyl phenyl sulphonamides as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-04-24 US disclosed
US-8163720-B2 Pyrrolidinyl phenyl sulphonamides as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-04-24 US disclosed