SCHEMBL26299072

SCHEMBL26299072

CC(=O)c1c(C)cnn1C

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
AHR P35869 1/20 0.36
HTT P42858 2/20 0.36
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2212203 0.83 L3MBTL1 (0.39) KMT2AMEN1AHRHTTSMN1; SMN2
SCHEMBL16963966 0.81 KMT2A (0.39) KMT2AMEN1AHRHTTPKM
SCHEMBL6608600 0.81 ALDH1A1 (0.42) KMT2AMEN1AHRHTTSMN1; SMN2
SCHEMBL2215634 0.78 CNR2 (0.47) KMT2AMEN1AHRHTT
SCHEMBL24553896 0.77 HTT (0.50) KMT2AHTTSMN1; SMN2LMNA
SCHEMBL8262559 0.77 HTT (0.53) KMT2AMEN1AHRHTTSMN1; SMN2
SCHEMBL23361708 0.76 KMT2A (0.36) KMT2AMEN1AHRHTTSMN1; SMN2
Hydrochloric Acid SCHEMBL23354295 0.75 KMT2A (0.35) KMT2AMEN1AHRHTTSMN1; SMN2
SCHEMBL2521960 0.75 KMT2A (0.48) KMT2ASMN1; SMN2LMNA
SCHEMBL23366891 0.74 SMN1; SMN2 (0.35) KMT2AMEN1AHRHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240174683-A1 MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-30 US disclosed
EP-4288437-A1 MAP4K1 INHIBITORS Bayer Aktiengesellschaft (DE) 2023-12-13 EP disclosed
WO-2023159307-A1 POLO-LIKE KINASE 4 (PLK4) INHIBITORS, PHARMACEUTICAL COMPOSITIONS, METHODS OF PREPARATION AND USES THEREOF REPARE THERAPEUTICS INC. (CA) 2023-08-31 WO disclosed
WO-2022167627-A1 MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2022-08-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174683-A1 MAP4K1 INHIBITORS MAP3K4, MAP4K4, MAP4K1 KMT2A 2250/4885MEN1 468/4885AHR 4407/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.