SCHEMBL26329520

SCHEMBL26329520

Cc1ncc(C(C)(C)N)cc1F

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
ALOX5AP P20292 1/20 0.35
VRK1 Q99986 1/20 0.33
PDE2A O00408 1/20 0.31
AGBL2 Q5U5Z8 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HTR1D P28221 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12169540 0.83 ALOX5AP (0.40) ALOX5APVRK1HTR1D
SCHEMBL7940202 0.83 AGBL2 (0.43) VRK1PDE2AAGBL2HDAC3HDAC1
SCHEMBL20089646 0.77 VRK1 (0.32) ALOX5APVRK1PDE2A
SCHEMBL26340897 0.76 VRK1 (0.37) VRK1AGBL2
SCHEMBL34471009 0.71 ALOX5AP (0.41) ALOX5APPDE2AHTR1D
SCHEMBL111804 0.70
SCHEMBL31153218 0.70
SCHEMBL254115 0.69
SCHEMBL29475255 0.69
SCHEMBL19996792 0.69 PDE2A (0.33) PIK3CAPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023158626-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF MERCK SHARP & DOHME LLC (US) 2023-08-24 WO disclosed