SCHEMBL2635745

SCHEMBL2635745

O=C(O)c1cccc(CC=NO)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 3/20 0.56
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HIF1A Q16665 1/20 0.46
ANPEP P15144 1/20 0.46
ENPEP Q07075 1/20 0.46
MEP1B Q16820 2/20 0.45
KMT2A Q03164 1/20 0.45
NR4A2 P43354 1/20 0.45
UNG P13051 1/20 0.44
MRGPRX4 Q96LA9 4/20 0.44
TP53 P04637 2/20 0.44
PKM P14618 2/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEP1A Q16819 1/20 0.44
RAB9A P51151 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28745456 1.00 FOLH1 (0.56) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL5070742 0.82 FOLH1 (0.63) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL17294137 0.81 FOLH1 (0.58) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL22227442 0.80 FOLH1 (0.61) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL529613 0.79 FOLH1 (0.56) FOLH1CYP2D6CYP2C9HIF1AANPEP
Benzene SCHEMBL28254095 0.79 FOLH1 (0.59) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL715984 0.79 FOLH1 (0.59) FOLH1CYP2D6CYP2C9HIF1AANPEP
SCHEMBL28393877 0.78 KMT2A (0.52) HIF1AANPEPENPEPKMT2ATP53
SCHEMBL4311596 0.76 ERN1 (0.47)
SCHEMBL8668550 0.76 UNG (0.62) FOLH1CYP2D6CYP2C9HIF1AANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920667-B Electrochemical preparation method of atta Lu Lunzhi 湖南大学 2024-06-21 CN claimed
CN-114920667-B Electrochemical preparation method of atta Lu Lunzhi 湖南大学 2024-06-21 CN disclosed
CN-114920667-A Electrochemical preparation method of astraglucol 湖南大学 2022-08-19 CN disclosed
EP-2585468-A1 PYRROLO- PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2013-05-01 EP disclosed
EP-2569313-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2013-03-20 EP disclosed
WO-2011163527-A1 PYRROLO- PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-12-29 WO disclosed
WO-2011143426-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-17 WO disclosed
CN-101665469-A Heterocyclic compounds useful as Nurrl activators NOVARTIS AG 2010-03-10 CN disclosed
CN-100475795-C Heterocyclic compounds useful as Nurr1 activators NOVARTIS AG (CH) 2009-04-08 CN disclosed
CN-101076703-A Compounds for nonsense inhibition and methods of use thereof PTC THERAPEUTICS INC (US) 2007-11-21 CN disclosed
CN-1747942-A Heterocyclic compounds useful as Nurr1 activators NOVARTIS AG (CH) 2006-03-15 CN disclosed