SCHEMBL263907

SCHEMBL263907

Fc1cc(Cl)cc(Br)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.37
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ERN1 O75460 1/20 0.34
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM1A O60341 2/20 0.31
KDM1B Q8NB78 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29363756 1.00 PDK2 (0.37) PDK2TSHRALDH1A1ERN1NPC1
SCHEMBL24602620 0.80 TSHR (0.47) TSHRALDH1A1HPGD
SCHEMBL12849942 0.80 TSHR (0.47) PDK2TSHRALDH1A1ERN1HPGD
SCHEMBL29948146 0.79 AKR1B1 (0.36) PDK2TSHRERN1NPC1RAB9A
SCHEMBL22165559 0.79 TSHR (0.35) PDK2TSHRERN1NPC1RAB9A
SCHEMBL29429741 0.79 TSHR (0.35) PDK2TSHRERN1NPC1RAB9A
SCHEMBL29428923 0.79 MAPT (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2KDM1A
SCHEMBL31619139 0.79 CYP3A4 (0.38) TSHRALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL20303393 0.79 MAPT (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2KDM1A
SCHEMBL3208926 0.79 CYP3A4 (0.38) TSHRALDH1A1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 147 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611700-B Preparation method of 1-bromo-2, 5-dichloro-3-fluorobenzene 辽宁东大光明化工科技有限责任公司 2024-06-14 CN claimed
CN-117430481-B Preparation method of 1-bromo-2, 5-dichloro-3-fluorobenzene 辽宁东大光明化工科技有限责任公司 2024-02-27 CN claimed
CN-117430481-A Preparation method of 1-bromo-2, 5-dichloro-3-fluorobenzene 辽宁东大光明化工科技有限责任公司 2024-01-23 CN claimed
CN-115611700-A Preparation method of 1-bromo-2,5-dichloro-3-fluorobenzene 辽宁东大光明化工科技有限责任公司 2023-01-17 CN claimed
US-20260042782-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 THERAPEUTICS, INC. (US) 2026-02-12 US disclosed
EP-4681715-A2 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 Therapeutics, Inc. (US) 2026-01-21 EP disclosed
US-20260007678-A1 COMBINATION OF ALLOSTERIC AND ORTHOSTERIC EGFR INHIBITORS FOR THE TREATMENT OF CANCER HOFFMANN-LA ROCHE INC. (US) 2026-01-08 US disclosed
EP-4076450-B1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 THERAPEUTICS INC (US) 2025-12-10 EP disclosed
US-12486290-B2 Isoindolinone and indazole compounds for the degradation of EGFR C4 THERAPEUTICS, INC. (US) 2025-12-02 US disclosed
US-12479849-B2 EGFR inhibitors for the treatment of cancer HOFFMANN-LA ROCHE INC. (US) 2025-11-25 US disclosed
US-20250289824-A1 EGFR INHIBITOR FOR THE TREATMENT OF CANCER HOFFMANN-LA ROCHE INC. (US) 2025-09-18 US disclosed
US-20250270234-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 THERAPEUTICS, INC. (US) 2025-08-28 US disclosed
WO-2007052123-A2 PYRAZINE DERIVATIVES AS SODIUM CHANNEL MODULATORS FOR THE TREATMENT OF PAIN PFIZER LIMITED (GB) 2007-05-10 WO disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP disclosed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO disclosed
US-20050239881-A1 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC 2005-10-27 US disclosed
US-20050239880-A1 Methods for treating retroviral infections ROCHE PALO ALTO LLC 2005-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050239880-A1 Methods for treating retroviral infections CCR5, CD38, CD4 PDK2 4668/4885TSHR 1735/4885ALDH1A1 428/4885
US-12486290-B2 Isoindolinone and indazole compounds for the degradation of EGFR EGFR, ERBB2, ERBB3 PDK2 1967/4885TSHR 2271/4885ALDH1A1 2283/4885
US-20260007678-A1 COMBINATION OF ALLOSTERIC AND ORTHOSTERIC EGFR INHIBITORS FOR THE TREATMENT OF CANCER EGFR, ERBB2, ERBB3 PDK2 3854/4885TSHR 108/4885ALDH1A1 3340/4885
US-20250270234-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR EGFR, ERBB2, ERBB3 PDK2 1967/4885TSHR 2271/4885ALDH1A1 2283/4885
US-20260042782-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR EGFR, ERBB2, ERBB3 PDK2 4452/4885TSHR 945/4885ALDH1A1 2446/4885
US-20250289824-A1 EGFR INHIBITOR FOR THE TREATMENT OF CANCER EGFR, ERBB2, ERBB4 PDK2 3599/4885TSHR 1160/4885ALDH1A1 3253/4885
US-12479849-B2 EGFR inhibitors for the treatment of cancer EGFR, ERBB2, ERBB3 PDK2 1398/4885TSHR 217/4885ALDH1A1 4090/4885
US-20050239881-A1 Non-nucleoside reverse transcriptase inhibitors RPP30, PNP, RTF1 PDK2 4422/4885TSHR 1773/4885ALDH1A1 2794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.