SCHEMBL2639463

SCHEMBL2639463

CCN(CC)C(=O)[C@@H]1CCCN(Cc2ccc(C(=O)NCCOC(=O)N(c3ccccc3-c3ccccc3)N3CC[CH]CC3)o2)C1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.46
POLB P06746 2/20 0.42
HTT P42858 1/20 0.41
ALDH1A1 P00352 5/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
AKT1 P31749 1/20 0.37
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272613 0.87 PDCD1 (0.38) POLBHTTALDH1A1RAB9AKMT2A
SCHEMBL2638612 0.86 KDM4E (0.50) KDM4EPOLBHTTALDH1A1MAPT
SCHEMBL2639950 0.83 CHRM2 (0.37) KDM4EPOLBALDH1A1RAB9AKMT2A
SCHEMBL6022003 0.83 KDM4E (0.50) KDM4EPOLBHTTALDH1A1MAPT
SCHEMBL4694436 0.80 NPC1 (0.38) HTTALDH1A1MAPTRAB9AKMT2A
SCHEMBL4693976 0.78 NPC1 (0.36) HTTALDH1A1RAB9AKMT2AHPGD
SCHEMBL6022004 0.78 POLB (0.43) KDM4EPOLBALDH1A1KMT2A
SCHEMBL1304570 0.76 CHRM3 (0.53)
SCHEMBL1304566 0.76 CHRM3 (0.53)
SCHEMBL5276784 0.73 EPHX2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4837653-B2 2011-12-14 JP claimed
JP-2008532922-A 2008-08-21 JP claimed
EP-1723114-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP claimed
WO-2005087738-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO claimed
EP-1723114-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP disclosed
WO-2005087738-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO disclosed