SCHEMBL26401518

SCHEMBL26401518

CS(=O)(=O)Nc1ccc(F)c(C(N)=O)c1F

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 1/20 0.43
FABP4 P15090 1/20 0.41
BRAF P15056 3/20 0.40
NEU3 Q9UQ49 1/20 0.40
MAPT P10636 1/20 0.39
ADRA2C P18825 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
MAP2K1 Q02750 4/20 0.38
EP300 Q09472 1/20 0.38
KAT2B Q92831 1/20 0.38
KAT8 Q9H7Z6 1/20 0.38
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.38
CA2 P00918 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13687178 0.85 MAP2K4 (0.42) MAP2K4FABP4BRAFMAPTEP300
SCHEMBL3529771 0.85 FABP4 (0.53) MAP2K4FABP4BRAFNEU3MAPT
SCHEMBL9931060 0.84 BRAF (0.49) MAP2K4BRAFMAP2K1CYP3A4CYP2C9
SCHEMBL26401647 0.83 CYP2C9 (0.42) FABP4BRAFMAP2K1CA2CYP3A4
SCHEMBL3019904 0.83 BRAF (0.51) FABP4BRAFMAP2K1CA2
SCHEMBL3526302 0.83 KDM4E (0.47) MAP2K4FABP4BRAFMAPTCYP2C9
SCHEMBL13687251 0.83 BRAF (0.43) MAP2K4FABP4BRAFMAPT
SCHEMBL13747696 0.81 BRAF (0.42) MAP2K4FABP4BRAFMAP2K1CYP3A4
SCHEMBL13719484 0.81 FABP4 (0.42) MAP2K4FABP4BRAFMAPT
SCHEMBL13687086 0.81 MAP2K4 (0.40) MAP2K4FABP4CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed