SCHEMBL26401647

SCHEMBL26401647

CC(C)S(=O)(=O)Nc1ccc(F)c(C(N)=O)c1F

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.42
CYP3A4 P08684 2/20 0.42
MAP2K1 Q02750 4/20 0.41
ACLY P53396 1/20 0.40
MLKL Q8NB16 1/20 0.40
BRAF P15056 6/20 0.39
FABP4 P15090 1/20 0.39
CYP2C19 P33261 3/20 0.39
CA2 P00918 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9930367 0.85 CYP2C9 (0.57) CYP2C9CYP3A4MAP2K1BRAFCYP2C19
SCHEMBL26401518 0.83 MAP2K4 (0.43) CYP2C9CYP3A4MAP2K1BRAFFABP4
SCHEMBL9931060 0.81 BRAF (0.49) CYP2C9CYP3A4MAP2K1BRAFCYP2C19
SCHEMBL10129554 0.80 ACLY (0.44) CYP2C9CYP3A4ACLYBRAFCYP2C19
SCHEMBL3019904 0.79 BRAF (0.51) MAP2K1BRAFFABP4CA2
SCHEMBL3017378 0.79 CYP2C19 (0.60) CYP2C9CYP3A4FABP4CYP2C19
SCHEMBL1492058 0.77 CYP3A4 (0.60) CYP2C9CYP3A4MAP2K1BRAFCYP2C19
SCHEMBL3026115 0.75 CYP2D6 (0.46) CYP3A4ACLYFABP4CA2
SCHEMBL1492020 0.75 FABP4 (0.48) BRAFFABP4
SCHEMBL3022486 0.74 FABP4 (0.50) ACLYBRAFFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed