SCHEMBL2640835

SCHEMBL2640835

NCC(O)Cc1ncc2[nH]cnc2n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
KDM4E B2RXH2 1/20 0.44
RXFP1 Q9HBX9 1/20 0.42
CDK2 P24941 2/20 0.36
PAK1 Q13153 1/20 0.35
CCNT1 O60563 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34
CCNH P51946 1/20 0.34
POLA1 P09884 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28839814 0.81 ALDH1A1 (0.46) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL5134319 0.79 ALDH1A1 (0.39) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL11200783 0.79 ALDH1A1 (0.58) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL28759590 0.78 ALDH1A1 (0.50) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL30020945 0.78 ALDH1A1 (0.49) ALDH1A1KDM4ERXFP1CDK2PAK1
Water SCHEMBL28488923 0.77 ALDH1A1 (0.56) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL5325201 0.77 SLC7A5 (0.47) ALDH1A1KDM4ERXFP1CDK2CCNT1
SCHEMBL23779416 0.75 ALDH1A1 (0.44) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL10694875 0.75 ALDH1A1 (0.46) ALDH1A1KDM4ERXFP1CDK2PAK1
Iodide SCHEMBL28673351 0.74 ALDH1A1 (0.53) ALDH1A1KDM4ERXFP1CDK2PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438068-A1 SUBSTITUTED 6-(2-HYDROXYBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THESE DERIVATIVES Univerzita Palackého v Olomouci (CZ) 2012-04-11 EP claimed
WO-2010139289-A1 SUBSTITUTED 6-(2-HYDROXYBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THESE DERIVATIVES UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2010-12-09 WO claimed