SCHEMBL26415728

SCHEMBL26415728

CC(=O)N1CC=C(S)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.47
NOTUM Q6P988 2/20 0.42
NAMPT P43490 1/20 0.38
PTAFR P25105 1/20 0.37
CYP1A2 P05177 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
MAPT P10636 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CASP6 P55212 1/20 0.33
GFER P55789 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
BAZ2B Q9UIF8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8386277 0.78 QDPR (0.53) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL8261115 0.78 QDPR (0.49) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL3307094 0.77 QDPR (0.50) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL18611164 0.76 QDPR (0.47) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL13804073 0.76 QDPR (0.47) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL14028045 0.75 PDK4 (0.50) NAMPTSMN1; SMN2
SCHEMBL11560724 0.74 QDPR (0.46) QDPRNOTUMPTAFRTSHRKMT2A
SCHEMBL13851469 0.74 QDPR (0.46) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL10412647 0.73 QDPR (0.45) QDPRNOTUMNAMPTPTAFRCYP1A2
SCHEMBL104852 0.73 QDPR (0.45) QDPRNOTUMNAMPTPTAFRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3675858-B1 IMIDAZO[1,5-A]PYRAZINE COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION OPTIKIRA LLC (US) 2023-04-26 EP disclosed