SCHEMBL2642001

SCHEMBL2642001

Clc1cccc(-c2cccc(-n3cnc4ccccc43)c2)c1

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 7/20 0.83
HTT P42858 1/20 0.58
HCAR1 Q9BXC0 1/20 0.49
HPGD P15428 2/20 0.48
CDK2 P24941 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29830083 0.91 FGFR1 (1.00) FGFR1HTTHCAR1HPGD
SCHEMBL27241663 0.91 FGFR1 (1.00) FGFR1HTTHCAR1HPGD
SCHEMBL4015486 0.88 HTT (0.71) FGFR1HTT
SCHEMBL2642019 0.82 FGFR1 (0.60) FGFR1HTT
SCHEMBL16158540 0.82 FGFR1 (0.83) FGFR1HTT
SCHEMBL3417304 0.82 HTT (0.78) FGFR1HTT
SCHEMBL2641988 0.81 FGFR1 (0.59) FGFR1HTT
SCHEMBL16158486 0.81 FGFR1 (0.59) FGFR1HTT
SCHEMBL13045092 0.80 FGFR1 (0.57) FGFR1HTT
SCHEMBL20180561 0.80 HTT (0.59) FGFR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563001-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1996-02-28 EP claimed
EP-0563001-A1 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1993-09-29 EP claimed
EP-0563001-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1996-02-28 EP disclosed
US-5360809-A Imidazole compounds and their use as calcium channel blockers NEUROSEARCH A/S (DK) 1994-11-01 US disclosed
EP-0563001-A1 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1993-09-29 EP disclosed