SCHEMBL2642011

SCHEMBL2642011

FC(F)(F)c1ccc2c(c1)ncn2-c1cccc(I)c1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.52
ALDH1A1 P00352 1/20 0.52
FGFR1 P11362 10/20 0.47
AURKA O14965 1/20 0.46
KDR P35968 1/20 0.46
AURKB Q96GD4 1/20 0.46
HTT P42858 1/20 0.46
F9 P00740 1/20 0.44
F10 P00742 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646769 0.88 HTT (0.59) HPGDALDH1A1FGFR1AURKAKDR
SCHEMBL19915930 0.86 FGFR1 (0.62) ALDH1A1FGFR1KDRHTT
SCHEMBL2666380 0.84 HPGD (0.52) HPGDALDH1A1FGFR1AURKAKDR
SCHEMBL2642078 0.84 FGFR1 (0.63) HPGDALDH1A1FGFR1AURKAKDR
SCHEMBL2641853 0.82 FGFR1 (0.65) HPGDALDH1A1FGFR1KDRHTT
SCHEMBL2641981 0.80 FGFR1 (0.56) HPGDALDH1A1FGFR1AURKAKDR
SCHEMBL1356729 0.80 FGFR1 (0.66) HPGDALDH1A1FGFR1AURKAKDR
SCHEMBL24119935 0.79 FGFR1 (0.69) FGFR1HTT
SCHEMBL2642101 0.79 HPGD (0.47) HPGDALDH1A1FGFR1AURKAKDR
Hydrochloric Acid SCHEMBL2641992 0.79 FGFR1 (0.54) HPGDALDH1A1FGFR1AURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0616807-B1 Benzimidazole useful in the treatment of central nervous system disorders NEUROSEARCH AS (DK) 1998-07-08 EP disclosed
US-5554632-A CENTRAL NERVOUS SYSTEM NEUROSEARCH A/S (DK) 1996-09-10 US disclosed
EP-0563001-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1996-02-28 EP disclosed
US-5360809-A Imidazole compounds and their use as calcium channel blockers NEUROSEARCH A/S (DK) 1994-11-01 US disclosed
EP-0616807-A1 Benzimidazole useful in the treatment of central nervous system disorders NEUROSEARCH A/S (DK) 1994-09-28 EP disclosed
EP-0563001-A1 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1993-09-29 EP disclosed