SCHEMBL2642064

SCHEMBL2642064

Cc1cccc(C)c1-c1ncccc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.54
NOS1 P29475 1/20 0.54
NOS2 P35228 1/20 0.54
CD44 P16070 1/20 0.46
PDK2 Q15119 1/20 0.46
CYP2A6 P11509 1/20 0.44
CYP3A4 P08684 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
PIK3CA P42336 1/20 0.41
METAP2 P50579 1/20 0.41
PLAU P00749 1/20 0.40
KMT2A Q03164 1/20 0.39
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PRMT5 O14744 1/20 0.38
CNR2 P34972 1/20 0.37
TGFBR1 P36897 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5208334 0.86 NOS3 (0.44) NOS3NOS1NOS2PDK2CYP2A6
SCHEMBL12320089 0.85 NOS3 (0.54) NOS3NOS1NOS2PDK2CYP2A6
SCHEMBL4436882 0.80 NOS3 (0.50) NOS3NOS1NOS2CD44CYP2A6
SCHEMBL29535498 0.79 HSP90AA1 (0.45) NOS3NOS1NOS2CYP3A4TDP1
SCHEMBL1083427 0.79 HSP90AA1 (0.45) NOS3NOS1NOS2CYP3A4TDP1
SCHEMBL2936584 0.78 NOS3 (0.44) NOS3NOS1NOS2CD44PDK2
SCHEMBL23175282 0.77 ALDH1A1 (0.48) TDP1LMNAPLAUKMT2AMAPT
SCHEMBL29625828 0.77 ALDH1A1 (0.48) TDP1LMNAPLAUKMT2AMAPT
SCHEMBL19463671 0.77 CD44 (0.50) NOS3NOS1NOS2CD44PDK2
SCHEMBL21681654 0.77 NOS3 (0.43) NOS3NOS1NOS2CD44PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563001-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1996-02-28 EP disclosed
US-5360809-A Imidazole compounds and their use as calcium channel blockers NEUROSEARCH A/S (DK) 1994-11-01 US disclosed
EP-0563001-A1 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1993-09-29 EP disclosed