SCHEMBL264279

SCHEMBL264279

CCN(CC)S(=O)(=O)c1cccc(Br)c1

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.69
SMN1; SMN2 Q16637 5/20 0.69
TSHR P16473 4/20 0.69
MAPT P10636 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
HSP90AA1 P07900 1/20 0.57
MAPK1 P28482 1/20 0.57
LMNA P02545 3/20 0.53
HTT P42858 1/20 0.52
GFER P55789 1/20 0.49
POLB P06746 1/20 0.48
KDM4E B2RXH2 1/20 0.48
ATM Q13315 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1511605 0.83 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL1511608 0.83 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL196097 0.81 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL9860335 0.80 ALDH1A1 (0.71) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL263946 0.79 RAB9A (0.54) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL31689487 0.79 RAB9A (0.54) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL938569 0.79 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL205074 0.79 SMN1; SMN2 (0.67) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL14376200 0.79 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2TSHRMAPTMEN1
SCHEMBL9321475 0.79 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2TSHRMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120035580-A Novel piperazinyl sulfonamides and their use as neuroprotective and/or neurorestorative agents 基因密码公司 2025-05-23 CN disclosed
WO-2024079351-A1 NOVEL PIPERAZINE-BASED SULFONAMIDES AND THEIR USE AS NEUROPROTECTIVE AND/OR NEURORESTORATIVE AGENTS GENECODE (EE) 2024-04-18 WO disclosed
EP-1951684-B1 BI-ARYL META-PYRIMIDINE INHIBITORS OF KINASES TARGEGEN INC (US) 2016-07-13 EP disclosed
US-8604042-B2 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2013-12-10 US disclosed
US-8138199-B2 Use of bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2012-03-20 US disclosed
US-8133900-B2 Use of bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2012-03-13 US disclosed
US-20110212077-A1 BI-ARYL META-PYRIMIDINE INHIBITORS OF KINASES TARGEGEN, INC. (US) 2011-09-01 US disclosed
US-7825246-B2 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2010-11-02 US disclosed
US-20090286789-A1 Bi-Aryl Meta-Pyrimidine Inhibitors of Kinases TARGEGEN, INC. (US) 2009-11-19 US disclosed
US-20090275582-A1 Bi-Aryl Meta-Pyrimidine Inhibitors of Kinases IMPACT BIOMEDICINES, INC. 2009-11-05 US disclosed
WO-2009103007-A2 STEROID HORMONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2009-08-20 WO disclosed
US-7528143-B2 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2009-05-05 US disclosed
US-20070259904-A1 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2007-11-08 US disclosed
US-20070191405-A1 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2007-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286789-A1 Bi-Aryl Meta-Pyrimidine Inhibitors of Kinases JAK2, TYK2, LTK ALDH1A1 3662/4885SMN1; SMN2 3530/4885TSHR 1587/4885
US-20070191405-A1 Bi-aryl meta-pyrimidine inhibitors of kinases JAK2, TYK2, JAK3 ALDH1A1 3235/4885SMN1; SMN2 4746/4885TSHR 1278/4885
US-20070259904-A1 Bi-aryl meta-pyrimidine inhibitors of kinases JAK2, TYK2, JAK3 ALDH1A1 3235/4885SMN1; SMN2 4746/4885TSHR 1278/4885
US-20090275582-A1 Bi-Aryl Meta-Pyrimidine Inhibitors of Kinases JAK2, TYK2, JAK3 ALDH1A1 3235/4885SMN1; SMN2 4746/4885TSHR 1278/4885
US-20110212077-A1 BI-ARYL META-PYRIMIDINE INHIBITORS OF KINASES JAK2, TYK2, JAK3 ALDH1A1 3235/4885SMN1; SMN2 4746/4885TSHR 1278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.