SCHEMBL2645280

SCHEMBL2645280

COC(=O)c1ccc(Oc2cc3nc(-c4ccccn4)[nH]c3cc2Oc2cccnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GCK P35557 16/20 0.52
CHEK2 O96017 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
RUNX1 Q01196 1/20 0.48
CBFB Q13951 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2645213 0.90 GCK (0.51) GCKCHEK2NPC1RAB9ARUNX1
SCHEMBL2646514 0.89 CHEK2 (0.60) GCKCHEK2NPC1RAB9A
SCHEMBL2645717 0.89 GCK (0.53) GCKCHEK2NPC1RAB9ARUNX1
SCHEMBL2645464 0.87 NPC1 (0.60) GCKNPC1RAB9ARUNX1CBFB
SCHEMBL2645586 0.84 GCK (0.59) GCKNPC1RAB9ARUNX1CBFB
SCHEMBL2646351 0.84 CHEK2 (0.55) GCKCHEK2NPC1RAB9ACBFB
SCHEMBL2645647 0.83 GCK (0.51) GCKNPC1RAB9ACBFB
SCHEMBL2647102 0.82 GCK (0.47) GCKNPC1RAB9ACBFB
SCHEMBL2644746 0.82 GCK (0.49) GCKNPC1RAB9ACBFB
SCHEMBL2645613 0.81 METAP2 (0.57) GCKCHEK2NPC1RAB9ARUNX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702919-B1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE MSD KK (JP) 2012-05-30 EP disclosed
EP-1702919-A1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-09-20 EP disclosed