SCHEMBL2646209

SCHEMBL2646209

O=[N+]([O-])c1cc(C(F)(F)F)cc([N+](=O)[O-])c1Nc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
HSP90AA1 P07900 1/20 0.55
ALDH1A1 P00352 6/20 0.51
TDP1 Q9NUW8 3/20 0.51
CYP3A4 P08684 2/20 0.51
HPGD P15428 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
HIF1A Q16665 1/20 0.51
TXNRD1 Q16881 1/20 0.51
TXNRD3 Q86VQ6 1/20 0.51
TXNRD2 Q9NNW7 1/20 0.51
KIF11 P52732 1/20 0.51
MAPK1 P28482 4/20 0.51
AKR1B1 P15121 2/20 0.51
AKR1C4 P17516 2/20 0.51
AKR1C3 P42330 2/20 0.51
AKR1C2 P52895 2/20 0.51
AKR1C1 Q04828 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646131 0.90 ALDH1A1 (0.56) MEN1KMT2AHSP90AA1ALDH1A1TDP1
SCHEMBL11590982 0.85 ALDH1A1 (0.56) MEN1KMT2AALDH1A1TDP1CYP3A4
SCHEMBL10527427 0.85 ALDH1A1 (0.53) MEN1KMT2AALDH1A1TDP1CYP3A4
SCHEMBL10799433 0.84 MEN1 (0.55) MEN1KMT2AHSP90AA1ALDH1A1TDP1
SCHEMBL13811262 0.82 MAPK1 (0.75) MEN1KMT2AALDH1A1TDP1CYP3A4
SCHEMBL10802521 0.81 MAPK1 (0.58) MEN1KMT2AALDH1A1TDP1CYP3A4
SCHEMBL10527474 0.80 MAPT (0.65) MEN1KMT2AALDH1A1CYP3A4HPGD
SCHEMBL10796892 0.80 KIF11 (0.58) MEN1KMT2AALDH1A1HPGDKIF11
SCHEMBL11156657 0.80 KMT2A (0.79) MEN1KMT2AHSP90AA1ALDH1A1TDP1
SCHEMBL11149199 0.80 MAPT (0.55) MEN1KMT2AHSP90AA1ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0616807-B1 Benzimidazole useful in the treatment of central nervous system disorders NEUROSEARCH AS (DK) 1998-07-08 EP disclosed
US-5554632-A CENTRAL NERVOUS SYSTEM NEUROSEARCH A/S (DK) 1996-09-10 US disclosed
US-5554630-A TREATING ANXIETY, CONVULSIONS AND SLEEP DISORDERS IN LIVING ANIMALS BY MODULATION OF THE BENZODIAZEPINE RECEPTOR OF THE CENTRAL NERVOUS SYSTEM WITH 1-/3-HETEROCYCLYLPHENYL/-BENZIMIDAZOLES NEUROSEARCH A/S (DK) 1996-09-10 US disclosed
EP-0616807-A1 Benzimidazole useful in the treatment of central nervous system disorders NEUROSEARCH A/S (DK) 1994-09-28 EP disclosed
US-4152460-A FUNGICIDES ELI LILLY AND COMPANY (US) 1979-05-01 US disclosed
US-4117167-A INSECTICIDES, ACARICIDES IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1978-09-26 US disclosed